# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4824939 | Binding | Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assay | Homo sapiens | 31 | ALA4823290 | single protein format | Scientific Literature | |
2. | ALA4824940 | Binding | Inhibition of PU-H71-FITC3 binding to recombinant N-terminal HSP90alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assay | Homo sapiens | 31 | ALA4823290 | single protein format | Scientific Literature | |
3. | ALA4824941 | Binding | Inhibition of PU-H71-FITC3 binding to recombinant N-terminal Grp94 (unknown origin) incubated for 2 hrs by fluorescence polarization assay | Homo sapiens | 31 | ALA4823290 | single protein format | Scientific Literature | |
4. | ALA4824942 | Binding | Selectivity index, ratio of IC50 for inhibition of HSP90alpha (unkown origin) to IC50 for inhibition of TRAP1 (unknown origin) | Homo sapiens | 30 | ALA4823290 | assay format | Scientific Literature | |
5. | ALA4824943 | Binding | Selectivity index, ratio of IC50 for inhibition of Grap94 (unkown origin) to IC50 for inhibition of TRAP1 (unknown origin) | Homo sapiens | 30 | ALA4823290 | assay format | Scientific Literature | |
6. | ALA4824944 | Binding | Inhibition of TRAP1 in human HeLa cells assessed as reduction in SDHB protein expression at 25 uM after 12 hrs by Western blotting analysis | Homo sapiens | 4 | ALA4823290 | cell-based format | Scientific Literature | |
7. | ALA4824946 | Binding | Inhibition of HSP90 in human HeLa cells assessed as reduction in HER2 protein expression at 25 uM after 12 hrs by Western blotting analysis | Homo sapiens | 5 | ALA4823290 | cell-based format | Scientific Literature | |
8. | ALA4824947 | Binding | Inhibition of HSP90alpha in human HeLa cells assessed as increase in HSP70 protein expression at 25 uM after 12 hrs by Western blotting analysis | Homo sapiens | 5 | ALA4823290 | cell-based format | Scientific Literature | |
9. | ALA4824948 | Binding | Inhibition of Grp94 in human HeLa cells assessed as reduction in cdk4 protein expression at 25 uM after 12 hrs by Western blotting analysis | Homo sapiens | 5 | ALA4823290 | cell-based format | Scientific Literature | |
10. | ALA4824949 | Binding | Inhibition of Grp94 in human HeLa cells assessed as reduction in HER2 protein expression at 25 uM after 12 hrs by Western blotting analysis | Homo sapiens | 5 | ALA4823290 | cell-based format | Scientific Literature | |
11. | ALA4824950 | Functional | Induction of apoptosis in human HeLa cells assessed as increase in cleaved caspase 3 protein expression at 25 uM after 12 hrs by Western blot analysis | Homo sapiens | 4 | ALA4823290 | cell-based format | Scientific Literature |