# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4824939 | B | Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assay | Homo sapiens | 31 | single protein format | Scientific Literature | ||
2. | ALA4824940 | B | Inhibition of PU-H71-FITC3 binding to recombinant N-terminal HSP90alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assay | Homo sapiens | 31 | single protein format | Scientific Literature | ||
3. | ALA4824941 | B | Inhibition of PU-H71-FITC3 binding to recombinant N-terminal Grp94 (unknown origin) incubated for 2 hrs by fluorescence polarization assay | Homo sapiens | 31 | single protein format | Scientific Literature | ||
4. | ALA4824942 | B | Selectivity index, ratio of IC50 for inhibition of HSP90alpha (unkown origin) to IC50 for inhibition of TRAP1 (unknown origin) | Homo sapiens | 30 | assay format | Scientific Literature | ||
5. | ALA4824943 | B | Selectivity index, ratio of IC50 for inhibition of Grap94 (unkown origin) to IC50 for inhibition of TRAP1 (unknown origin) | Homo sapiens | 30 | assay format | Scientific Literature | ||
6. | ALA4824944 | B | Inhibition of TRAP1 in human HeLa cells assessed as reduction in SDHB protein expression at 25 uM after 12 hrs by Western blotting analysis | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
7. | ALA4824946 | B | Inhibition of HSP90 in human HeLa cells assessed as reduction in HER2 protein expression at 25 uM after 12 hrs by Western blotting analysis | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
8. | ALA4824947 | B | Inhibition of HSP90alpha in human HeLa cells assessed as increase in HSP70 protein expression at 25 uM after 12 hrs by Western blotting analysis | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
9. | ALA4824948 | B | Inhibition of Grp94 in human HeLa cells assessed as reduction in cdk4 protein expression at 25 uM after 12 hrs by Western blotting analysis | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
10. | ALA4824949 | B | Inhibition of Grp94 in human HeLa cells assessed as reduction in HER2 protein expression at 25 uM after 12 hrs by Western blotting analysis | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
11. | ALA4824950 | F | Induction of apoptosis in human HeLa cells assessed as increase in cleaved caspase 3 protein expression at 25 uM after 12 hrs by Western blot analysis | Homo sapiens | 4 | cell-based format | Scientific Literature |