# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4824071 | Binding | Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assay | Homo sapiens | 35 | ALA4823258 | single protein format | Scientific Literature | |
2. | ALA4824072 | Binding | Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assay | Homo sapiens | 35 | ALA4823258 | single protein format | Scientific Literature | |
3. | ALA4824073 | Binding | Selectivity ratio of IC50 for His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate to IC50 for His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assay | Homo sapiens | 35 | ALA4823258 | assay format | Scientific Literature | |
4. | ALA4824084 | Binding | Inhibition of CBP/EP300 in human MM1.S cells assessed as perturbation of IRF4/Myc axis at 2.5 uM incubated for 2 hrs by immunoblot analysis | Homo sapiens | 4 | ALA4823258 | cell-based format | Scientific Literature |