| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4810421 | B | Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintillation counting method | Homo sapiens | 39 | single protein format | Scientific Literature | ||
| 2. | ALA4810423 | B | Inhibition of recombinant full length human Aurora A using LRRASLG as substrate incubated for 40 mins in presence of [gamma-33ATP] by radiometric scintillation counting method | Homo sapiens | 17 | single protein format | Scientific Literature | ||
| 3. | ALA4810424 | B | Inhibition of recombinant human IGF-1R (959 to end residues) using KKKSPGEYVNIEF as substrate incubated for 40 mins in presence of [gamma-33ATP] by radiometric scintillation counting method | Homo sapiens | 9 | single protein format | Scientific Literature | ||
| 4. | ALA4810425 | B | Inhibition of recombinant human FAK (411 to 686 residues) at 1 uM using EEEEYEEEEEEYY as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 5. | ALA4810426 | B | Inhibition of recombinant human ZIPK (1 to 290 residues) at 1 uM using KKLNRTLSFAEPG substrate incubated for 40 mins in presence of [gamma33P]ATP by scintillation counting based radiometry assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA4810427 | B | Inhibition of recombinant human CHK2 (5 to end residues) at 1 uM using KKKVSRSGLYRSPSMPENLNRPR as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 7. | ALA4810428 | B | Inhibition of recombinant human TRKA (440 to end residues) at 1 uM using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by scintillation counting based radiometry assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA4810429 | B | Inhibition of recombinant human ZIPK (1 to 290 residues) using KKLNRTLSFAEPG substrate incubated for 40 mins in presence of [gamma33P]ATP by scintillation counting based radiometry assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA4810430 | B | Inhibition of recombinant human CHK2 (5 to end residues) using KKKVSRSGLYRSPSMPENLNRPR as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA4810431 | B | Inhibition of recombinant human FAK (411 to 686 residues) using EEEEYEEEEEEYY as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA4810432 | B | Inhibition of recombinant human TRKA (440 to end residues) using KKKSPGEYVNIEFG as substrate incubated for 40 mins in presence of [gamma33P]ATP by scintillation counting based radiometry assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA4810433 | B | Selectivity index, ratio of IC50 for inhibition of human FAK to IC50 for inhibition of human GRK6 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 13. | ALA4810434 | B | Selectivity index, ratio of IC50 for inhibition of human ZIPK to IC50 for inhibition of human GRK6 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA4810435 | B | Selectivity index, ratio of IC50 for inhibition of human TRKA to IC50 for inhibition of human GRK6 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA4810436 | B | Selectivity index, ratio of IC50 for inhibition of human CHK2 to IC50 for inhibition of human GRK6 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 16. | ALA4810437 | B | Inhibition of recombinant human JAK2 (808 to end residues) using KTFCGTPEYLAPE as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scintillation counting analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA4810438 | B | Inhibition of recombinant human LTK (450 to end residues) at 1 uM using GEEPLYWSFPAKK as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scintillation counting analysis relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA4810439 | B | Inhibition of human GRK1 using casein as substrate in presence of [gamma33P]ATP by radiometric hotspot kinase assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 19. | ALA4810440 | B | Inhibition of human GRK2 using casein as substrate in presence of [gamma33P]ATP by radiometric hotspot kinase assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 20. | ALA4810441 | B | Inhibition of human GRK3 using casein as substrate in presence of [gamma33P]ATP by radiometric hotspot kinase assay | Homo sapiens | 3 | single protein format | Scientific Literature |
The page will load shortly, Thanks for your patience!