| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4834988 | B | Inhibition of recombinant SAE (unknown origin) assessed as reduction in transfer of SUMO1 to UBC9 using SUMO1 as a substrate in presence of ATP at Km concentration by HTRF assay | Homo sapiens | 60 | protein complex format | Scientific Literature | ||
| 2. | ALA4834989 | B | Inhibition of recombinant UAE (unknown origin) in presence of ATP at Km concentration by HTRF assay | Homo sapiens | 60 | assay format | Scientific Literature | ||
| 3. | ALA4834990 | B | Inhibition of recombinant NAE (unknown origin) in presence of ATP at Km concentration by HTRF assay | Homo sapiens | 60 | protein complex format | Scientific Literature | ||
| 4. | ALA4834998 | B | Inhibition of SAE in human HCT116 cells assessed as reduction in redistribution of SUMO2/3 proteins from nucleus to cytosol incubated for 4 hrs by immunofluorescence assay | Homo sapiens | 59 | cell-based format | Scientific Literature | ||
| 5. | ALA4835003 | B | Inhibition of SAE in human HCT116 cells assessed as redistribution of SUMO2/3 proteins from nucleus to cytosol preincubated for 2 hrs followed by compound washout and measured immediately by immunofluorescence assay | Homo sapiens | 25 | cell-based format | Scientific Literature | ||
| 6. | ALA4835004 | B | Inhibition of SAE in human HCT116 cells assessed as redistribution of SUMO2/3 proteins from nucleus to cytosol preincubated for 2 hrs followed by compound washout and measured after 8 hrs by immunofluorescence assay | Homo sapiens | 25 | cell-based format | Scientific Literature |
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