| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4836630 | Binding | Inhibition of 6His-Thr-BRD4 (1 to 477 residues) BD2 domain Y390A mutant (unknown origin) incubated for 30 mins by TR-FRET assay | Homo sapiens | 40 | ALA4834466 | single protein format | Scientific Literature | |
| 2. | ALA4836631 | Binding | Inhibition of 6His-Thr-BRD4 (1 to 477 residues) BD1 domain (unknown origin) incubated for 30 mins by TR-FRET assay | Homo sapiens | 40 | ALA4834466 | single protein format | Scientific Literature | |
| 3. | ALA4836632 | Physicochemical | Lipophilicity, logD of compound at pH 7.4 | 40 | ALA4834466 | small-molecule physicochemical format | Scientific Literature | ||
| 4. | ALA4836633 | Physicochemical | Solubility by CLND assay | 40 | ALA4834466 | small-molecule physicochemical format | Scientific Literature | ||
| 5. | ALA4836636 | Binding | Selectivity index, ratio of pIC50 for binding affinity to 6His-Thr-BRD4 (1 to 477 residues) BD1 domain (unknown origin) to pIC50 for binding affinity to 6His-Thr-BRD4 (1 to 477 residues) BD2 domain Y390A mutant (unknown origin) | Homo sapiens | 40 | ALA4834466 | assay format | Scientific Literature |
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