| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4827441 | Binding | Displacement of Alexa Fluor 647 labelled ligand from 6His-tagged BRD4 BD1/BD2 Y390A mutant (1 to 477 residue) (unknown origin) measured after 30 mins by TR-FRET assay | Homo sapiens | 43 | ALA4825709 | single protein format | Scientific Literature | |
| 2. | ALA4827442 | Binding | Displacement of Alexa Fluor 647 labelled ligand from 6His-tagged BRD4 BD2/BD1 Y97A mutant (1 to 477 residue) (unknown origin) measured after 30 mins by TR-FRET assay | Homo sapiens | 43 | ALA4825709 | single protein format | Scientific Literature | |
| 3. | ALA4827443 | Binding | Selectivity ratio of IC50 for 6His-tagged BRD4 BD1/BD2 Y390A mutant (1 to 477 residue) (unknown origin) to IC50 for 6His-tagged BRD4 BD2/BD1 Y97A mutant (1 to 477 residue) (unknown origin) | Homo sapiens | 43 | ALA4825709 | assay format | Scientific Literature | |
| 4. | ALA4827450 | Physicochemical | Lipophilicity, logD of compound at pH 7.4 by HPLC analysis | 41 | ALA4825709 | small-molecule physicochemical format | Scientific Literature | ||
| 5. | ALA4827451 | ADME | Apparent permeability of compound at pH 7.4 by artificial membrane permeability assay | 43 | ALA4825709 | assay format | Scientific Literature |
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