| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4829376 | B | Inhibition of human 20S proteasome LMP2 using Ac-PAL-AMC as fluorogenic substrate measured every minute for 1 hr by fluorescence assay | Homo sapiens | 20 | single protein format | Scientific Literature | ||
| 2. | ALA4829377 | B | Inhibition of human 20S proteasome Y using Ac-nLPnLD-AMC as fluorogenic substrate measured every minute for 1 hr by fluorescence assay | Homo sapiens | 20 | assay format | Scientific Literature | ||
| 3. | ALA4829378 | B | Inhibition of human 20S proteasome LMP7 using Ac-ANW-AMC as fluorogenic substrate measured every minute for 1 hr by fluorescence assay | Homo sapiens | 20 | single protein format | Scientific Literature | ||
| 4. | ALA4829379 | B | Inhibition of human 20S proteasome X using Ac-WLA-AMC as fluorogenic substrate measured every minute for 1 hr by fluorescence assay | Homo sapiens | 20 | assay format | Scientific Literature | ||
| 5. | ALA4829383 | B | Inhibition of human 20S proteasome LMP2 activity in human RPMI-8226 cells using Ac-PAL-AMC as fluorogenic substrate incubated for 72 hrs by fluorescence assay | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 6. | ALA4829384 | B | Inhibition of human 20S proteasome LMP2 activity in human RPMI-8226 cells overexpressing ABCB1 using Ac-PAL-AMC as fluorogenic substrate incubated for 72 hrs by fluorescence assay | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 7. | ALA4829385 | B | Selectivity index, ratio of IC50 for inhibition of human 20S proteasome LMP2 activity in human RPMI-8226 cells overexpressing ABCB1 to IC50 for inhibition of human 20S proteasome LMP2 activity in human RPMI-8226 cells | Homo sapiens | 5 | cell-based format | Scientific Literature |
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