| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA686311 | B | Inhibitory concentration was determined against human glycogen synthase kinase-3 alpha | 74 | single protein format | Scientific Literature | |||
| 2. | ALA930273 | B | Inhibition of recombinant GSK3-beta | 151 | single protein format | Scientific Literature | |||
| 3. | ALA3988182 | F | GSK PKIS2: Screen against O. lienalis microfilariae, single point, at 3.1uM to assess reduction in motility. Compounds were also tested for cytotoxicity against Rhesus Monkey LLCMK2 cells. A score was assigned as follows: Score 3 = Good activity, 100 % motility reduction; Score 2 = Marginal/moderate activity, 50-99% motility reduction; Score 1 = Inactive, <50% motility reduction; Score 0 = Cytotoxic. | Onchocerca lienalis | 486 | cell-based format | Published Kinase Inhibitor Set 2 | ||
| 4. | ALA5252697 | B | Inhibition of NEK1 (unknown origin) at 1 uM relative to control | Homo sapiens | 61 | single protein format | Scientific Literature | ||
| 5. | ALA5252698 | B | Inhibition of NEK2 (unknown origin) at 1 uM relative to control | Homo sapiens | 43 | single protein format | Scientific Literature | ||
| 6. | ALA5252699 | B | Inhibition of NEK3 (unknown origin) at 1 uM relative to control | Homo sapiens | 40 | single protein format | Scientific Literature | ||
| 7. | ALA5252700 | B | Inhibition of NEK4 (unknown origin) at 1 uM relative to control | Homo sapiens | 46 | single protein format | Scientific Literature | ||
| 8. | ALA5252701 | B | Inhibition of NEK5 (unknown origin) at 1 uM relative to control | Homo sapiens | 40 | single protein format | Scientific Literature | ||
| 9. | ALA5252702 | B | Inhibition of NEK6 (unknown origin) at 1 uM relative to control | Homo sapiens | 42 | single protein format | Scientific Literature | ||
| 10. | ALA5252703 | B | Inhibition of NEK7 (unknown origin) at 1 uM relative to control | Homo sapiens | 42 | single protein format | Scientific Literature | ||
| 11. | ALA5252704 | B | Inhibition of NEK9 (unknown origin) at 1 uM relative to control | Homo sapiens | 42 | single protein format | Scientific Literature | ||
| 12. | ALA5252705 | B | Inhibition of NEK10 (unknown origin) at 1 uM relative to control | Homo sapiens | 43 | single protein format | Scientific Literature | ||
| 13. | ALA5252706 | B | Inhibition of NEK11 (unknown origin) at 1 uM relative to control | Homo sapiens | 40 | single protein format | Scientific Literature |
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