| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5042559 | B | Inhibition of full length human HDAC8 using FAM-labeled acetylated peptide as substrate by electrophoretic mobility shift assay | Homo sapiens | 15 | ALA5042469 | single protein format | Scientific Literature | |
| 2. | ALA5042560 | B | Inhibition of full length human HDAC11 using FAM-labeled acetylated peptide as substrate by electrophoretic mobility shift assay | Homo sapiens | 15 | ALA5042469 | single protein format | Scientific Literature | |
| 3. | ALA5042561 | B | Inhibition of full length human HDAC5 using FAM-labeled acetylated peptide as substrate by electrophoretic mobility shift assay | Homo sapiens | 1 | ALA5042469 | single protein format | Scientific Literature | |
| 4. | ALA5042562 | B | Inhibition of full length human HDAC6 using FAM-labeled acetylated peptide as substrate by electrophoretic mobility shift assay | Homo sapiens | 21 | ALA5042469 | single protein format | Scientific Literature | |
| 5. | ALA5042563 | A | Stability in mouse plasma assessed as compound remaining measured after 30 mins | Mus musculus | 1 | ALA5042469 | cell-free format | Scientific Literature | |
| 6. | ALA5042564 | B | Inhibition of full length human HDAC4 using FAM-labeled acetylated peptide as substrate by electrophoretic mobility shift assay | Homo sapiens | 1 | ALA5042469 | single protein format | Scientific Literature | |
| 7. | ALA5042565 | B | Inhibition of full length human HDAC7 using FAM-labeled acetylated peptide as substrate by electrophoretic mobility shift assay | Homo sapiens | 1 | ALA5042469 | single protein format | Scientific Literature | |
| 8. | ALA5042566 | B | Inhibition of full length human HDAC2 using FAM-labeled acetylated peptide as substrate by electrophoretic mobility shift assay | Homo sapiens | 1 | ALA5042469 | single protein format | Scientific Literature | |
| 9. | ALA5042567 | B | Inhibition of full length human HDAC1 using FAM-labeled acetylated peptide as substrate by electrophoretic mobility shift assay | Homo sapiens | 1 | ALA5042469 | single protein format | Scientific Literature | |
| 10. | ALA5042568 | B | Inhibition of full length human HDAC3 using FAM-labeled acetylated peptide as substrate by electrophoretic mobility shift assay | Homo sapiens | 15 | ALA5042469 | single protein format | Scientific Literature | |
| 11. | ALA5042569 | B | Binding affinity to human HDAC6 by jump dilution assay | Homo sapiens | 1 | ALA5042469 | single protein format | Scientific Literature | |
| 12. | ALA5042570 | B | Inhibition of full length human HDAC9 using FAM-labeled acetylated peptide as substrate by electrophoretic mobility shift assay | Homo sapiens | 1 | ALA5042469 | single protein format | Scientific Literature | |
| 13. | ALA5042571 | B | Inhibition of full length human HDAC10 using FAM-labeled acetylated peptide as substrate by electrophoretic mobility shift assay | Homo sapiens | 1 | ALA5042469 | single protein format | Scientific Literature | |
| 14. | ALA5042572 | B | Inhibition of full length human HDAC6 using FAM-labeled acetylated peptide as substrate without preincubation by mass spectrometry analysis | Homo sapiens | 1 | ALA5042469 | single protein format | Scientific Literature | |
| 15. | ALA5042573 | B | Inhibition of full length human HDAC6 preincubated for 3 hrs by mass spectrometry analysis | Homo sapiens | 1 | ALA5042469 | single protein format | Scientific Literature | |
| 16. | ALA5042574 | B | Inhibition of HDAC6 (unknown origin) by fluorescence polarization assay | Homo sapiens | 1 | ALA5042469 | single protein format | Scientific Literature | |
| 17. | ALA5042575 | B | Inhibition of HDAC6 in human MV4-11 cells assessed as increase in acetylation of alpha tubulin at 0.25 uM by Western blot analysis | Homo sapiens | 2 | ALA5042469 | cell-based format | Scientific Literature | |
| 18. | ALA5042576 | B | Inhibition of HDAC6 in human AML cells assessed as acetylation of histone H3K27 accumulation at 0.75 to 1.00 uM by western blotting analysis | Homo sapiens | 2 | ALA5042469 | cell-based format | Scientific Literature | |
| 19. | ALA5042577 | B | Inhibition of HDAC6 in human MM.1S cells assessed as acetylation of histone H3K27 accumulation at 0.75 to 1.00 uM by western blotting analysis | Homo sapiens | 2 | ALA5042469 | cell-based format | Scientific Literature | |
| 20. | ALA5042578 | B | Inhibition of HDAC6 in human HeLa cells assessed as acetylation of alpha tubulin accumulation at 0.1 uM by DAPI staining based immunofluorescent assay | Homo sapiens | 2 | ALA5042469 | cell-based format | Scientific Literature |
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