| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5042436 | B | Displacement of [3H]-Citalopram from NET (unknown origin) expressed in HEK cell membrane incubated for 2 hrs by liquid scintillation counter analysis | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 2. | ALA5042437 | B | Displacement of [3H]-Citalopram from SERT receptor (unknown origin) expressed in HEK cell membrane incubated for 2 hrs by liquid scintillation counter analysis | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 3. | ALA5042438 | B | Displacement of [3H]-Citalopram from NMDA receptor (unknown origin) expressed in HEK cell membrane incubated for 2 hrs by liquid scintillation counter analysis | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 4. | ALA5042439 | B | Displacement of [3H]-Citalopram from sigma-2 receptor (unknown origin) expressed in HEK cell membrane incubated for 2 hrs by liquid scintillation counter analysis | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 5. | ALA5042440 | B | Displacement of [3H]-Citalopram from sigma-1 receptor (unknown origin) expressed in HEK cell membrane incubated for 2 hrs by liquid scintillation counter analysis | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 6. | ALA5042441 | P | Aqueous solubility of compound in universal buffer at pH 7.4 at 100 uM incubated for 1.5 hrs under shaking condition by LC-MS/MS analysis | 14 | small-molecule physicochemical format | Scientific Literature | |||
| 7. | ALA5042442 | P | Aqueous solubility of compound in universal buffer at pH 3 at 100 uM incubated for 1.5 hrs under shaking condition by LC-MS/MS analysis | 14 | small-molecule physicochemical format | Scientific Literature | |||
| 8. | ALA5042443 | B | Inhibition of human SERT receptor expressed in human HEK293 cells assessed as inhibition of substrate transport measured after 1 hr by flourescence based plate reader assay | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 9. | ALA5042444 | B | Inhibition of human NET expressed in human HEK293 cells assessed as inhibition of substrate transport measured after 1 hr by flourescence based plate reader assay | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 10. | ALA5042445 | T | Inhibition of human ERG at 10 uM measured after 15 mins by plate reader method relative to control | Homo sapiens | 5 | assay format | Scientific Literature | ||
| 11. | ALA5042446 | A | Stability in human liver microsomes assesses as intrinsic clearance at 10 uM measured upto 120 mins by LC-MS/MS analysis | Homo sapiens | 14 | microsome format | Scientific Literature | ||
| 12. | ALA5042447 | A | Stability in human liver microsomes assessed as half life at 10 uM measured upto 120 mins by LC-MS/MS analysis | Homo sapiens | 14 | microsome format | Scientific Literature | ||
| 13. | ALA5042448 | A | Apparent permeability in dog MDCK-MDR1 cells from apical to basal side measured after 30 to 120 mins by LC-MS analysis | Canis lupus familiaris | 7 | cell-based format | Scientific Literature | ||
| 14. | ALA5042449 | A | Apparent permeability in dog MDCK-MDR1 cells from basal to apical side measured after 30 to 120 mins by LC-MS analysis | Canis lupus familiaris | 7 | cell-based format | Scientific Literature | ||
| 15. | ALA5042450 | A | Efflux ratio of apparent permeability across basolateral to apical side over apical to basolateral side in dog MDCK-MDR1 cells measured after 30 to 120 mins by LC-MS analysis | Canis lupus familiaris | 7 | cell-based format | Scientific Literature | ||
| 16. | ALA5042451 | A | Cmax in Sprague-Dawley rat plasma at 2.5 mg/kg, po measured after 24 hrs by LC-MS/MS analysis | Rattus norvegicus | 6 | organism-based format | Scientific Literature | ||
| 17. | ALA5042452 | A | Cmax in Sprague-Dawley rat brain at 2.5 mg/kg, po measured after 24 hrs by LC-MS/MS analysis | Rattus norvegicus | 6 | organism-based format | Scientific Literature | ||
| 18. | ALA5042453 | A | AUC in Sprague-Dawley rat plasma at 2.5 mg/kg, po measured after 24 hrs by LC-MS/MS analysis | Rattus norvegicus | 6 | organism-based format | Scientific Literature | ||
| 19. | ALA5042454 | A | AUC in Sprague-Dawley rat brain at 2.5 mg/kg, po measured after 24 hrs by LC-MS/MS analysis | Rattus norvegicus | 6 | organism-based format | Scientific Literature | ||
| 20. | ALA5042455 | A | Unbound concentration in Sprague-Dawley rat plasma at 20 uM measured by NMR analysis | Rattus norvegicus | 6 | cell-free format | Scientific Literature |
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