| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5044758 | B | Agonist activity at PPARalpha (unknown origin) | Homo sapiens | 47 | ALA5042526 | single protein format | Scientific Literature | |
| 2. | ALA5044759 | B | Agonist activity at PPARdelta (unknown origin) | Homo sapiens | 47 | ALA5042526 | single protein format | Scientific Literature | |
| 3. | ALA5044760 | B | Agonist activity at PPARgamma (unknown origin) | Homo sapiens | 47 | ALA5042526 | single protein format | Scientific Literature | |
| 4. | ALA5044761 | B | Agonist activity at PPARalpha (unknown origin) assessed as maximal activation at 10 nM relative to GW7647 | Homo sapiens | 40 | ALA5042526 | single protein format | Scientific Literature | |
| 5. | ALA5044762 | B | Agonist activity at PPARdelta (unknown origin) assessed as maximal activation at 10 nM relative to GW501516 | Homo sapiens | 39 | ALA5042526 | single protein format | Scientific Literature | |
| 6. | ALA5044763 | B | Agonist activity at PPARgamma (unknown origin) assessed as maximal activation at 10 nM relative to Rosiglitazone | Homo sapiens | 29 | ALA5042526 | single protein format | Scientific Literature | |
| 7. | ALA5044767 | B | Selectivity ratio of EC50 for PPARgamma (unknown origin) to EC50 of PPARdelta (unknown origin) | Homo sapiens | 2 | ALA5042526 | protein format | Scientific Literature | |
| 8. | ALA5044768 | B | Selectivity ratio of EC50 for PPARgamma (unknown origin) to EC50 of PPARalpha (unknown origin) | Homo sapiens | 2 | ALA5042526 | assay format | Scientific Literature | |
| 9. | ALA5044769 | B | Potency index, ratio of EC50 for IVA337 to EC50 for test compound for agonist activity at PPARalpha (unknown origin) | Homo sapiens | 1 | ALA5042526 | single protein format | Scientific Literature | |
| 10. | ALA5044770 | B | Potency index, ratio of EC50 for IVA337 to EC50 for test compound for agonist activity at PPARdelta (unknown origin) | Homo sapiens | 1 | ALA5042526 | single protein format | Scientific Literature | |
| 11. | ALA5044848 | A | Microsomal stability in human liver microsomes assessed as terminal elimination half life at 1 uM measured upto 60 mins by LC-MS/MS-11 analysis | Homo sapiens | 9 | ALA5042526 | microsome format | Scientific Literature | |
| 12. | ALA5044849 | A | Intrinsic clearance in human liver microsomes at 1 uM measured upto 60 mins by LC-MS/MS-11 analysis | Homo sapiens | 9 | ALA5042526 | microsome format | Scientific Literature |
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