| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5030191 | B | Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 1 hr by scintillation counting method | Rattus norvegicus | 8 | ALA5029183 | cell membrane format | Scientific Literature | |
| 2. | ALA5030192 | B | Displacement of [3H]DPDPE from DOR in Wistar rat brain membranes measured after 3 hrs by scintillation counting method | Rattus norvegicus | 8 | ALA5029183 | cell membrane format | Scientific Literature | |
| 3. | ALA5030193 | B | Displacement of [3H]-U69593 from KOR in Wistar rat brain membranes measured after 1 hr by scintillation counting method | Rattus norvegicus | 8 | ALA5029183 | cell membrane format | Scientific Literature | |
| 4. | ALA5030194 | B | Selectivity index, ratio of Ki for displacement of [3H]DPDPE from DOR in Wistar rat brain membranes to Ki for displacement of [3H]DAMGO from MOR in Wistar rat brain membranes | Rattus norvegicus | 8 | ALA5029183 | cell membrane format | Scientific Literature | |
| 5. | ALA5030195 | B | Selectivity index, ratio of Ki for displacement of [3H]-U69593 from KOR in Wistar rat brain membranes to Ki for displacement of [3H]DAMGO from MOR in Wistar rat brain membranes | Rattus norvegicus | 8 | ALA5029183 | cell membrane format | Scientific Literature | |
| 6. | ALA5030196 | F | Inhibition of electric-field induced guinea pig ileum contraction | Cavia porcellus | 8 | ALA5029183 | tissue-based format | Scientific Literature | |
| 7. | ALA5030197 | F | Inhibition of electric-field induced mouse vas deferens contraction | Mus musculus | 8 | ALA5029183 | tissue-based format | Scientific Literature | |
| 8. | ALA5030198 | F | Agonist activity at mu-opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 15 mins by ELISA | Homo sapiens | 8 | ALA5029183 | cell-based format | Scientific Literature | |
| 9. | ALA5030199 | F | Agonist activity at mu-opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 15 mins by ELISA relative to control | Homo sapiens | 8 | ALA5029183 | cell-based format | Scientific Literature | |
| 10. | ALA5030200 | F | Agonist activity at delta-opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 15 mins by ELISA | Homo sapiens | 6 | ALA5029183 | cell-based format | Scientific Literature | |
| 11. | ALA5030201 | F | Agonist activity at kappa-opioid receptor (unknown origin) expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 15 mins by ELISA | Homo sapiens | 6 | ALA5029183 | cell-based format | Scientific Literature | |
| 12. | ALA5030202 | A | Metabolic stability in Kunming mouse brain assessed as half life measured upto 480 mins by RP-HPLC analysis | Mus musculus | 8 | ALA5029183 | tissue-based format | Scientific Literature | |
| 13. | ALA5030203 | A | Metabolic stability in Kunming mouse serum assessed as half life measured upto 480 mins by RP-HPLC analysis | Mus musculus | 8 | ALA5029183 | cell-free format | Scientific Literature | |
| 14. | ALA5030204 | P | Octanol/buffer distribution coefficient, log D of the compound at pH 7.4 by RP-HPLC analysis | 8 | ALA5029183 | small-molecule physicochemical format | Scientific Literature |
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