| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5034352 | B | Inhibition of human NatD using H4-8 peptide substrate at Km value and AcCoA measured after 30 min incubation by fluorescence assay | Homo sapiens | 10 | ALA5034000 | single protein format | Scientific Literature | |
| 2. | ALA5034353 | B | Inhibition of human NatD using H4-8 peptide substrate at 4 times Km value and AcCoA measured after 30 min incubation by fluorescence assay | Homo sapiens | 10 | ALA5034000 | single protein format | Scientific Literature | |
| 3. | ALA5034354 | B | Inhibition of human NatD using H4-8 peptide substrate at Km value and AcCoA by Morrison's quadratic equation analysis | Homo sapiens | 10 | ALA5034000 | single protein format | Scientific Literature | |
| 4. | ALA5034355 | B | Non-competitive inhibition of human NatD using various concentration of [14C]acetyl-CoA and fixed human H4 peptide as substrate measured after 13 mins radioactive assay | Homo sapiens | 1 | ALA5034000 | single protein format | Scientific Literature | |
| 5. | ALA5034356 | B | Competitive inhibition of human NatD using various concentration of human H4 peptide and fixed [14C]acetyl-CoA as substrate measured after 13 mins radioactive assay | Homo sapiens | 1 | ALA5034000 | single protein format | Scientific Literature | |
| 6. | ALA5034357 | B | Non-competitive inhibition of human NatD using various concentration of [14C]acetyl-CoA and fixed human H4 peptide as substrate assessed as Km of substrate measured after 13 mins radioactive assay | Homo sapiens | 1 | ALA5034000 | single protein format | Scientific Literature | |
| 7. | ALA5034358 | B | Competitive inhibition of human NatD using various concentration of human H4 peptide and fixed [14C]acetyl-CoA as substrate assessed as Km of substrate measured after 13 mins radioactive assay | Homo sapiens | 1 | ALA5034000 | single protein format | Scientific Literature | |
| 8. | ALA5034359 | B | Inhibition of human NatB using AcCoA and H4 peptide as substrate at 10 uM incubated for 12 min at room temperature | Homo sapiens | 2 | ALA5034000 | assay format | Scientific Literature | |
| 9. | ALA5034360 | B | Selectivity ratio of inhibition of human NatB to inhibition of human NatD | Homo sapiens | 1 | ALA5034000 | assay format | Scientific Literature | |
| 10. | ALA5034361 | B | Selectivity ratio of inhibition of human NatC to inhibition of human NatD | Homo sapiens | 1 | ALA5034000 | assay format | Scientific Literature | |
| 11. | ALA5034362 | B | Selectivity ratio of inhibition of human NatE to inhibition of human NatD | Homo sapiens | 1 | ALA5034000 | assay format | Scientific Literature | |
| 12. | ALA5034363 | B | Selectivity ratio of inhibition of human PCAF to inhibition of human NatD | Homo sapiens | 1 | ALA5034000 | assay format | Scientific Literature | |
| 13. | ALA5034364 | B | Selectivity ratio of inhibition of human NatA to inhibition of human NatD | Homo sapiens | 1 | ALA5034000 | assay format | Scientific Literature | |
| 14. | ALA5034365 | B | Selectivity ratio of inhibition of human MOF to inhibition of human NatD | Homo sapiens | 1 | ALA5034000 | assay format | Scientific Literature | |
| 15. | ALA5034366 | B | Inhibition of human NatC using AcCoA and H4 peptide as substrate at 10 uM incubated for 12 min at room temperature | Homo sapiens | 2 | ALA5034000 | assay format | Scientific Literature | |
| 16. | ALA5034367 | B | Inhibition of human NatE using AcCoA and H4 peptide as substrate at 10 uM incubated for 12 min at room temperature | Homo sapiens | 2 | ALA5034000 | single protein format | Scientific Literature | |
| 17. | ALA5034368 | B | Inhibition of human PCAF using AcCoA and H4 peptide as substrate at 10 uM incubated for 12 min at room temperature | Homo sapiens | 2 | ALA5034000 | single protein format | Scientific Literature | |
| 18. | ALA5034369 | A | Drug uptake in digitonin treated human HCT116 cells measured at 100 uM after 2 hrs of incubation by MALDI-MS | Homo sapiens | 2 | ALA5034000 | cell-based format | Scientific Literature | |
| 19. | ALA5034370 | B | Thermal stabilization of human NatD using digitonin treated human HCT-116 cell lysate assessed as increase in melting apparent aggregation temperature at 100 uM compound treated cells and lysed after 2 hrs by CETSA | Homo sapiens | 2 | ALA5034000 | subcellular format | Scientific Literature | |
| 20. | ALA5034371 | B | Inhibition of human NatA using AcCoA and H4 peptide as substrate at 1 uM incubated for 12 min at room temperature relative to control | Homo sapiens | 1 | ALA5034000 | assay format | Scientific Literature |
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