| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5044758 | B | Agonist activity at PPARalpha (unknown origin) | Homo sapiens | 47 | ALA5042526 | single protein format | Scientific Literature | |
| 2. | ALA5044759 | B | Agonist activity at PPARdelta (unknown origin) | Homo sapiens | 47 | ALA5042526 | single protein format | Scientific Literature | |
| 3. | ALA5044760 | B | Agonist activity at PPARgamma (unknown origin) | Homo sapiens | 47 | ALA5042526 | single protein format | Scientific Literature | |
| 4. | ALA5044761 | B | Agonist activity at PPARalpha (unknown origin) assessed as maximal activation at 10 nM relative to GW7647 | Homo sapiens | 40 | ALA5042526 | single protein format | Scientific Literature | |
| 5. | ALA5044762 | B | Agonist activity at PPARdelta (unknown origin) assessed as maximal activation at 10 nM relative to GW501516 | Homo sapiens | 39 | ALA5042526 | single protein format | Scientific Literature | |
| 6. | ALA5044763 | B | Agonist activity at PPARgamma (unknown origin) assessed as maximal activation at 10 nM relative to Rosiglitazone | Homo sapiens | 29 | ALA5042526 | single protein format | Scientific Literature | |
| 7. | ALA5044767 | B | Selectivity ratio of EC50 for PPARgamma (unknown origin) to EC50 of PPARdelta (unknown origin) | Homo sapiens | 2 | ALA5042526 | protein format | Scientific Literature | |
| 8. | ALA5044768 | B | Selectivity ratio of EC50 for PPARgamma (unknown origin) to EC50 of PPARalpha (unknown origin) | Homo sapiens | 2 | ALA5042526 | assay format | Scientific Literature | |
| 9. | ALA5044771 | B | Agonist activity at human PPARalpha transfected in Cos7 cells co-expressing pBIND and pGL4.35 Gal4 UAS Luc reporter plasmid by measuring luciferase activity incubated for 16 hrs by luciferase reporter gene assay | Homo sapiens | 1 | ALA5042526 | cell-based format | Scientific Literature | |
| 10. | ALA5044772 | B | Agonist activity at human PPARdelta transfected in Cos7 cells co-expressing with pBIND and pGL4.35 Gal4 UAS Luc reporter plasmid by measuring luciferase activity incubated for 16 hrs by luciferase reporter gene assay | Homo sapiens | 1 | ALA5042526 | cell-based format | Scientific Literature | |
| 11. | ALA5044773 | B | Agonist activity at human PPARgamma transfected in Cos7 cells co-expressing with pBIND and pGL4.35 Gal4 UAS Luc reporter plasmid by measuring luciferase activity incubated for 16 hrs by luciferase reporter gene assay | Homo sapiens | 1 | ALA5042526 | cell-based format | Scientific Literature | |
| 12. | ALA5044774 | B | Agonist activity at mouse PPARalpha transfected in Cos7 cells co-expressing with pBIND and pGL4.35 Gal4 UAS Luc reporter plasmid by measuring luciferase activity incubated for 16 hrs by luciferase reporter gene assay | Mus musculus | 1 | ALA5042526 | cell-based format | Scientific Literature | |
| 13. | ALA5044775 | B | Agonist activity at mouse PPARdelta in Cos7 cells transfected with pBIND and pGL4.35 Gal4 UAS Luc reporter plasmid by measuring luciferase activity incubated for 16 hrs by luciferase reporter gene assay | Mus musculus | 1 | ALA5042526 | cell-based format | Scientific Literature | |
| 14. | ALA5044776 | B | Agonist activity at mouse PPARgamma in Cos7 cells transfected with pBIND and pGL4.35 Gal4 UAS Luc reporter plasmid by measuring luciferase activity incubated for 16 hrs by luciferase reporter gene assay | Mus musculus | 1 | ALA5042526 | cell-based format | Scientific Literature | |
| 15. | ALA5044777 | B | Agonist activity against PPARalpha/delta (unknown origin) assessed as upregulation of ACADVL mRNA expression in human HepG2 cells incubated for 12 hrs by RT-PCR analysis | Homo sapiens | 1 | ALA5042526 | cell-based format | Scientific Literature | |
| 16. | ALA5044778 | B | Agonist activity against PPARalpha/delta (unknown origin) assessed as upregulation of PDK4 mRNA expression in human HepG2 cells incubated for 12 hrs by RT-PCR analysis | Homo sapiens | 1 | ALA5042526 | cell-based format | Scientific Literature | |
| 17. | ALA5044779 | B | Agonist activity against PPARalpha/delta (unknown origin) assessed as upregulation of CPT1A mRNA expression in human HepG2 cells incubated for 12 hrs by RT-PCR analysis | Homo sapiens | 1 | ALA5042526 | cell-based format | Scientific Literature | |
| 18. | ALA5044780 | B | Agonist activity against PPARalpha/delta (unknown origin) assessed as upregulation of ACADVL mRNA expression in human HepG2 cells at 8 nM incubated for 12 hrs by RT-PCR analysis | Homo sapiens | 1 | ALA5042526 | cell-based format | Scientific Literature | |
| 19. | ALA5044781 | B | Agonist activity against PPARalpha/delta (unknown origin) assessed as upregulation of PDK4 mRNA expression in human HepG2 cells at 8 nM incubated for 12 hrs by RT-PCR analysis | Homo sapiens | 1 | ALA5042526 | cell-based format | Scientific Literature | |
| 20. | ALA5044782 | B | Agonist activity against PPARalpha/delta (unknown origin) assessed as upregulation of CPT1A mRNA expression in human HepG2 cells at 8 nM incubated for 12 hrs by RT-PCR analysis | Homo sapiens | 1 | ALA5042526 | cell-based format | Scientific Literature |
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