| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5037539 | B | Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assay | Homo sapiens | 17 | single protein format | Scientific Literature | ||
| 2. | ALA5037540 | B | Inhibition of CHK2 (unknown origin) at 3 uM by Z-lyte assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 3. | ALA5037541 | B | Inhibition of LRRK2 (unknown origin) at 3 uM by ADAPTA assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 4. | ALA5037542 | F | Antiproliferative activity against human CAL-51 cells assessed as inhibition of cell proliferation measured after 3 days by Cell Titer-Glo luminescence based assay | Homo sapiens | 17 | cell-based format | Scientific Literature | ||
| 5. | ALA5037543 | P | Kinetic solubility of compound in PBS at pH 7.4 at 200 uM incubated for 24 hrs by UPLC/MS analysis | 17 | small-molecule physicochemical format | Scientific Literature | |||
| 6. | ALA5037544 | A | Clearance in rat at 2 mg/kg, iv | Rattus norvegicus | 17 | organism-based format | Scientific Literature | ||
| 7. | ALA5037545 | A | Inhibition of CYP3A4 in human liver microsomes using ketoconazole as substrate incubated for 5 mins in presence of NADPH by LC-MS/MS analysis | Homo sapiens | 19 | microsome format | Scientific Literature | ||
| 8. | ALA5037546 | B | Inhibition of CHK2 (unknown origin) by Z-lyte assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA5037547 | B | Inhibition of LRRK2 (unknown origin) by ADAPTA assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA5037548 | B | Inhibition of LRRK2 G2019S mutant (unknown origin) by ADAPTA assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA5037549 | B | Inhibition of JNK1 (unknown origin) by Z-lyte assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA5037550 | B | Inhibition of JNK2 (unknown origin) by Z-lyte assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA5037551 | B | Inhibition of MAPKAPK3 (unknown origin) by Z-lyte assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA5037552 | B | Inhibition of SRC N1 (unknown origin) by Z-lyte assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA5037553 | B | Inhibition of TSSK2 (unknown origin) by Z-lyte assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA5037554 | B | Inhibition of TSSK1 (unknown origin) by Z-lyte assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA5037555 | B | Selectivity index, ratio of IC50 for inhibition of CHK2 (unknown origin) to IC50 for inhibition of TTK (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 18. | ALA5037556 | B | Selectivity ratio of IC50 for inhibition of LRRK2 (unknown origin) to IC50 for inhibition of TTK (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 19. | ALA5037557 | B | Selectivity ratio of IC50 for inhibition of LRRK2 G2019S mutant (unknown origin) to IC50 for inhibition of TTK (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 20. | ALA5037558 | B | Selectivity ratio of IC50 for inhibition of JNK1 (unknown origin) to IC50 for inhibition of TTK (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature |
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