| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5043811 | B | Inhibition of GST-tagged DCN1 (unknown origin) using AcUBE2M1-21 incubated for 30 mins by HTRF assay | Homo sapiens | 62 | ALA5042502 | single protein format | Scientific Literature | |
| 2. | ALA5043812 | F | Effect on Ang II-induced in Cul4B neddylation in mouse cardiac fibroblast at 1 uM preincubated for 2 hrs followed by Ang-II stimulation and further incubated for 24 hrs by western blot analysis | Mus musculus | 1 | ALA5042502 | cell-based format | Scientific Literature | |
| 3. | ALA5043813 | T | Cytotoxicity against Sprague-Dawley rat cardiac fibroblast incubated for 24 hrs by MTT assay | Rattus norvegicus | 1 | ALA5042502 | cell-based format | Scientific Literature | |
| 4. | ALA5043814 | B | Binding affinity to extracellular DCN1 (unknown origin) assessed as dissociation constant incubated for upto 180 secs by label-free biolayer interferometry assay | Homo sapiens | 1 | ALA5042502 | single protein format | Scientific Literature | |
| 5. | ALA5043815 | B | Binding affinity to DCN1 (unknown origin) assessed as change in entropy by MM-PBSA method | Homo sapiens | 3 | ALA5042502 | single protein format | Scientific Literature | |
| 6. | ALA5043816 | B | Binding affinity to DCN1 (unknown origin) assessed as Gibbs free energy change by MM-PBSA method | Homo sapiens | 3 | ALA5042502 | single protein format | Scientific Literature | |
| 7. | ALA5043817 | B | Binding affinity to DCN1 (unknown origin) assessed as inhibitory constant | Homo sapiens | 2 | ALA5042502 | single protein format | Scientific Literature | |
| 8. | ALA5043818 | B | Binding affinity to DCN2 (unknown origin) assessed as inhibitory constant | Homo sapiens | 2 | ALA5042502 | single protein format | Scientific Literature | |
| 9. | ALA5043819 | B | Binding affinity to DCN3 (unknown origin) assessed as inhibitory constant | Homo sapiens | 2 | ALA5042502 | single protein format | Scientific Literature | |
| 10. | ALA5043820 | B | Binding affinity to DCN4 (unknown origin) assessed as inhibitory constant | Homo sapiens | 2 | ALA5042502 | single protein format | Scientific Literature | |
| 11. | ALA5043821 | B | Binding affinity to DCN5 (unknown origin) assessed as inhibitory constant | Homo sapiens | 2 | ALA5042502 | single protein format | Scientific Literature | |
| 12. | ALA5043822 | B | Inhibition of NEDD8-UBC12 (unknown origin) interaction in presence of ATP at 100 uM by densitometry | Homo sapiens | 1 | ALA5042502 | assay format | Scientific Literature | |
| 13. | ALA5043823 | B | Inhibition of intracellular DCN1 in Sprague-Dawley rat cardiac fibroblast measured between 42 to 62 degC at 10 uM incubated for 5 hrs by cellular thermal shift assay | Rattus norvegicus | 1 | ALA5042502 | cell-based format | Scientific Literature | |
| 14. | ALA5043824 | B | Inhibition of DCN1 in Sprague-Dawley rat cardiac fibroblast assessed as suppression in DCN1-UBC12 interaction by measuring reduction in UBC12 level at 10 uM incubated for 5 hrs co-incubated with DCN1 antibody by co-immunoprecipitation pull down assay | Rattus norvegicus | 2 | ALA5042502 | cell-based format | Scientific Literature | |
| 15. | ALA5043825 | B | Inhibition of DCN1 in Ang II-treated Sprague-Dawley rat cardiac fibroblast assessed as inhibition of cell proliferation preincubated for 2 hrs followed by Ang-II stimulation and further incubated for 24 hrs by MTT assay | Rattus norvegicus | 1 | ALA5042502 | cell-based format | Scientific Literature | |
| 16. | ALA5043826 | T | Cytotoxicity against Sprague-Dawley rat cardiac fibroblast by MTT assay | Rattus norvegicus | 9 | ALA5042502 | cell-based format | Scientific Literature | |
| 17. | ALA5043827 | B | Inhibition of DCN1 in TGF-beta-treated Sprague-Dawley rat cardiac fibroblast assessed as inhibition of cell proliferation at 0.1 to 3 uM preincubated for 2 hrs followed by TGF-beta stimulation and further incubated for 24 hrs by MTT assay | Rattus norvegicus | 1 | ALA5042502 | cell-based format | Scientific Literature | |
| 18. | ALA5043828 | B | Inhibition of DCN1 in Ang II-treated Sprague-Dawley rat cardiac fibroblast assessed as decrease in cell migration preincubated for 2 hrs followed by Ang-II stimulation and further incubated for 24 hrs by scratch wound healing assay based microscopy | Rattus norvegicus | 1 | ALA5042502 | cell-based format | Scientific Literature | |
| 19. | ALA5043829 | B | Inhibition of DCN1 in Ang II-treated Sprague-Dawley rat cardiac fibroblast assessed as inhibited cell migration at 0.1 to 3 uM incubated for 24 hrs stained with crystal violet by transwell migration assay | Rattus norvegicus | 1 | ALA5042502 | cell-based format | Scientific Literature | |
| 20. | ALA5043830 | F | Inhibition of differentiation of Ang II-induced mouse cardiac fibroblast to myofibroblast assessed as decrease in alpha-SMA expression levels at 1 uM preincubated for 2 hrs followed by Ang-II stimulation and further incubated for 24 hrs by immunofluorescence assay | Mus musculus | 1 | ALA5042502 | cell-based format | Scientific Literature |
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