| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5043484 | B | Protac activity at human CDK12/CycK in human Bel-7402 cells assessed as degradation of CDK12 at 3 uM measured after 24 hrs by Western blotting assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 2. | ALA5043485 | B | Inhibition of human CDK12 (696 to 1082 residues) /cyclinK (1 to 300 residues) using ac-YSPTSPpSYSPTSFpS-YSPTSPpSY-[PEG2]-RR-amid peptide as substrate in presence of ATP measured after 2 hrs by ADP-Glo kinase assay | Homo sapiens | 7 | protein complex format | Scientific Literature | ||
| 3. | ALA5043486 | B | Protac activity at human CDK12/CycK in human MDA-MB-231 cells assessed as degradation of CDK12 at 3 uM measured after 24 hrs by Western blotting assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 4. | ALA5043514 | B | Inhibition of human N-terminal FLAG-tagged CDK13 (600 to 1100 residues) using GST-tagged CTD as substrate at 3 uM for 2 hrs by western blot analysis | Homo sapiens | 1 | single protein format | Scientific Literature |
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