| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5069389 | B | Reverse ITC (compound as receptor). Domain start/stop: V50-P350 | Homo sapiens | 1 | ALA5069381 | single protein format | EUbOPEN Chemogenomic Library | |
| 2. | ALA5167572 | B | Inhibition of human N-terminal His-tagged/ TEV cleavage fused DRAK1 (39 to 369 residues) expressed in Escherichia coli assessed as change in enthalpy by isothermal titration calorimetry | Homo sapiens | 2 | ALA5154923 | assay format | Scientific Literature | |
| 3. | ALA5167573 | B | Binding affinity to human N-terminal His-tagged/ TEV cleavage fused DRAK1 (39 to 369 residues) expressed in Escherichia coli assessed as change in melting temperature at 10 uM by SYPRO orange dye based DSF assay | Homo sapiens | 7 | ALA5154923 | assay format | Scientific Literature | |
| 4. | ALA5167574 | B | Binding affinity to wild type full length human CK2alpha1 (1 to 391 residues) expressed in mammalian expression system assessed as change in melting temperature at 10 uM by SYPRO orange dye based DSF assay | Homo sapiens | 7 | ALA5154923 | assay format | Scientific Literature | |
| 5. | ALA5167575 | B | Binding affinity to wild type full length human CK2alpha2 (1 to 350 residues) expressed in mammalian expression system assessed as change in melting temperature by SYPRO orange dye based DSF assay | Homo sapiens | 7 | ALA5154923 | assay format | Scientific Literature | |
| 6. | ALA5167576 | B | Binding affinity to wild type full length human DRAK2 (1 to 372 residues) expressed in bacterial expression system assessed as change in melting temperature by SYPRO orange dye based DSF assay | Homo sapiens | 23 | ALA5154923 | assay format | Scientific Literature | |
| 7. | ALA5167577 | B | Binding affinity to human N-terminal His-tagged/ TEV cleavage fused DRAK1 (39 to 369 residues) expressed in Escherichia coli by isothermal titration calorimetry | Homo sapiens | 2 | ALA5154923 | assay format | Scientific Literature | |
| 8. | ALA5167578 | B | Inhibition of human N-terminal His-tagged/ TEV cleavage fused DRAK1 (39 to 369 residues) expressed in Escherichia coli using KKLNRTLSFAEPG peptide as substrate in presence of [gamma-33P]ATP by radiometric based scintillation proximity assay | Homo sapiens | 4 | ALA5154923 | assay format | Scientific Literature | |
| 9. | ALA5167579 | B | Inhibition of human CK2alpha1 using RRRDDDSDDD peptide as substrate in presence of [gamma-33P]ATP by radiometric based scintillation proximity assay | Homo sapiens | 1 | ALA5154923 | single protein format | Scientific Literature | |
| 10. | ALA5167580 | B | Inhibition of human CK2alpha2 using RRRDDDSDDD peptide as substrate in presence of [gamma-33P]ATP by radiometric based scintillation proximity assay | Homo sapiens | 1 | ALA5154923 | assay format | Scientific Literature | |
| 11. | ALA5167581 | B | Inhibition of human N-terminal His-tagged/ TEV cleavage fused DRAK1 (39 to 369 residues) transfected in HEK293T cells using NanoBRET NanoGlo as substrate incubated for 2 hrs by NanoBRET assay | Homo sapiens | 7 | ALA5154923 | cell-based format | Scientific Literature | |
| 12. | ALA5167582 | B | Inhibition of CK2alpha1(unknown origin) transfected in HEK293T cells using NanoBRET NanoGlo as substrate incubated for 2 hrs by NanoBRET assay | Homo sapiens | 1 | ALA5154923 | cell-based format | Scientific Literature | |
| 13. | ALA5167583 | B | Inhibition of CK2alpha2 (unknown origin) transfected in HEK293T cells using NanoBRET NanoGlo as substrate incubated for 2 hrs by NanoBRET assay | Homo sapiens | 1 | ALA5154923 | cell-based format | Scientific Literature | |
| 14. | ALA5167584 | B | Inhibition of GAK (unknown origin) transfected in HEK293T cells using NanoBRET NanoGlo as substrate incubated for 2 hrs by NanoBRET assay | Homo sapiens | 1 | ALA5154923 | cell-based format | Scientific Literature | |
| 15. | ALA5167585 | B | Inhibition of BIKE (unknown origin) transfected in HEK293T cells using NanoBRET NanoGlo as substrate incubated for 2 hrs by NanoBRET assay | Homo sapiens | 1 | ALA5154923 | cell-based format | Scientific Literature | |
| 16. | ALA5167586 | B | Inhibition of DRAK2 (unknown origin) transfected in HEK293T cells using NanoBRET NanoGlo as substrate incubated for 2 hrs by NanoBRET assay | Homo sapiens | 1 | ALA5154923 | cell-based format | Scientific Literature | |
| 17. | ALA5167587 | B | Binding affinity to BIKE (unknown origin) assessed as change in melting temperature at 10 uM by SYPRO orange dye based DSF assay | Homo sapiens | 1 | ALA5154923 | single protein format | Scientific Literature | |
| 18. | ALA5167588 | B | Binding affinity to AAK1 (unknown origin) assessed as change in melting temperature at 10 uM by SYPRO orange dye based DSF assay | Homo sapiens | 1 | ALA5154923 | single protein format | Scientific Literature | |
| 19. | ALA5167589 | B | Inhibition of human N-terminal His-tagged/ TEV cleavage fused DRAK1 (39 to 369 residues) expressed in Escherichia coli assessed as change in entropy by isothermal titration calorimetry | Homo sapiens | 2 | ALA5154923 | assay format | Scientific Literature | |
| 20. | ALA5167590 | B | Inhibition of human N-terminal His-tagged/ TEV cleavage fused DRAK1 (39 to 369 residues) expressed in Escherichia coli assessed as gibbs free energy change by isothermal titration calorimetry | Homo sapiens | 2 | ALA5154923 | assay format | Scientific Literature |
The page will load shortly, Thanks for your patience!