| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5036641 | B | Binding affinity to human hexa-His tagged MPS1 (515 to 795 residue) expressed in Escherichia coli BL2I-DE3 cells assessed as change in melting temperature by thermal shift assay | Homo sapiens | 24 | cell-based format | Scientific Literature | ||
| 2. | ALA5036642 | F | Growth inhibition of human MDA-MB-231 cells measured after 5 days by CellTiter-Glo assay | Homo sapiens | 25 | cell-based format | Scientific Literature | ||
| 3. | ALA5036643 | B | Inhibition of human hexa-His tagged MPS1 (515 to 795 residue) expressed in Escherichia coli BL2I-DE3 cells incubated for 4 hrs in presence of ATP by ADP-glo luminescence assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 4. | ALA5036644 | A | Metabolic stability in human liver microsomes assessed as compound remaining after 30 mins | Homo sapiens | 4 | microsome format | Scientific Literature | ||
| 5. | ALA5036645 | A | Half life in ICR mouse at 10 mg/kg, po | Mus musculus | 4 | organism-based format | Scientific Literature | ||
| 6. | ALA5036646 | A | Cmax in ICR mouse at 10 mg/kg, po | Mus musculus | 4 | organism-based format | Scientific Literature | ||
| 7. | ALA5036647 | A | AUC in ICR mouse at 10 mg/kg, po | Mus musculus | 4 | organism-based format | Scientific Literature | ||
| 8. | ALA5036648 | A | Oral bioavailability in ICR mouse at 10 mg/kg | Mus musculus | 4 | organism-based format | Scientific Literature |
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