# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA5158756 | B | Activation of human ABCG2-mediated ATPase activity preincubated for 2 mins followed by ATP addition at 1 M and measured after 20 mins by colorimetric assay relative to control | Homo sapiens | 29 | ALA5154735 | single protein format | Scientific Literature | |
2. | ALA5158757 | B | Activation of human ABCG2-mediated ATPase activity preincubated for 2 mins followed by ATP addition at 100 nM and measured after 20 mins by colorimetric assay relative to control | Homo sapiens | 18 | ALA5154735 | single protein format | Scientific Literature | |
3. | ALA5158759 | B | Activation of human ABCG2-mediated ATPase activity preincubated for 2 mins followed by ATP addition and measured after 20 mins by colorimetric assay | Homo sapiens | 10 | ALA5154735 | single protein format | Scientific Literature | |
4. | ALA5158761 | B | Inhibition of human ABCG2 in human R5 cells assessed as inhibition of mitoxantrone efflux at 10 uM measured by flow cytometric analysis relative to control | Homo sapiens | 11 | ALA5154735 | cell-based format | Scientific Literature | |
5. | ALA5158762 | B | Inhibition of human ABCG2 in human R5 cells assessed as inhibition of mitoxantrone efflux measured by flow cytometric analysis | Homo sapiens | 3 | ALA5154735 | cell-based format | Scientific Literature | |
6. | ALA5158763 | B | Binding affinity towards human adenosine A3 receptor | Homo sapiens | 29 | ALA5154735 | single protein format | Scientific Literature | |
7. | ALA5158764 | B | Binding affinity towards mouse adenosine A3 receptor | Mus musculus | 1 | ALA5154735 | single protein format | Scientific Literature | |
8. | ALA5158765 | B | Binding affinity towards human adenosine A1 receptor | Homo sapiens | 2 | ALA5154735 | single protein format | Scientific Literature | |
9. | ALA5158766 | B | Binding affinity towards human adenosine A2A receptor | Homo sapiens | 2 | ALA5154735 | single protein format | Scientific Literature | |
10. | ALA5158767 | B | Binding affinity towards human kappa opioid receptor | Homo sapiens | 1 | ALA5154735 | single protein format | Scientific Literature | |
11. | ALA5233319 | B | Binding affinity to human adenosine A3 receptor assessed as inhibition constant | Homo sapiens | 4 | ALA5233204 | single protein format | Scientific Literature | |
12. | ALA5233324 | B | Binding affinity to mouse adenosine A3 receptor assessed as inhibition constant | Mus musculus | 4 | ALA5233204 | single protein format | Scientific Literature | |
13. | ALA5233340 | B | Binding affinity to DOR (unknown origin) | Homo sapiens | 2 | ALA5233204 | single protein format | Scientific Literature | |
14. | ALA5233341 | B | Binding affinity to KOR (unknown origin) | Homo sapiens | 2 | ALA5233204 | single protein format | Scientific Literature | |
15. | ALA5233342 | B | Activation of human KOR assessed as beta-arrestin 2 recruitment at 30 uM by PathHunter enzyme fragment complementation assay relative to control | Homo sapiens | 2 | ALA5233204 | single protein format | Scientific Literature | |
16. | ALA5233343 | B | Binding affinity to MOR (unknown origin) | Homo sapiens | 2 | ALA5233204 | single protein format | Scientific Literature |