| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5125528 | B | Inhibition of mouse HDAC6 expressed in human HEK-293T cells using fluorescent peptide Ac-KGLGK(Ac)-MCA as substrate preincubated for 10 mins followed by substrate addition and measured after 1 hr by fluorogenic assay | Mus musculus | 8 | cell-based format | Scientific Literature | ||
| 2. | ALA5125529 | B | Inhibition of human HDAC1 expressed in human HEK-293T cells using fluorescent peptide RHKKAc as substrate preincubated for 10 mins followed by substrate addition and measured after 1 hr by fluorogenic assay | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 3. | ALA5125530 | B | Inhibition of human HDAC4 using fluorescent peptide Boc-Lys(trifluoroacetyl)-AMC as substrate preincubated for 10 mins followed by substrate addition and measured after 30 mins by fluorogenic assay | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 4. | ALA5125531 | B | Selectivity ratio of IC50 for inhibition of human HDAC1 expressed in human HEK-293T cells using fluorescent peptide RHKKAc as substrate to IC50 for inhibition of mouse HDAC6 expressed in human HEK-293T cells using fluorescent peptide Ac-KGLGK(Ac)-MCA as substrate | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 5. | ALA5125532 | B | Selectivity ratio of IC50 for inhibition of human HDAC4 using fluorescent peptide Boc-Lys(trifluoroacetyl)-AMC as substrate to IC50 for inhibition of mouse HDAC6 expressed in human HEK-293T cells using fluorescent peptide Ac-KGLGK(Ac)-MCA as substrate | Homo sapiens | 6 | cell-based format | Scientific Literature |
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