| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5167881 | B | Inhibition of PRMT1 (unknown origin) using histone H4 (1 to 21 residues) peptide as substrate incubated for 210 mins in presence of SAM by AlphaLISA assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 2. | ALA5167883 | F | Antiproliferation activity against human A-375 cells assessed as cell growth inhibition incubated for 5 days by CCK-8 assay | Homo sapiens | 16 | cell-based format | Scientific Literature | ||
| 3. | ALA5167884 | A | Metabolic stability in human liver microsomes assessed as clearance incubated for 10 mins measured up to 60 mins in presence of NADPH by LC-MS/MS analysis | Homo sapiens | 11 | microsome format | Scientific Literature | ||
| 4. | ALA5167885 | A | Metabolic stability in human liver microsomes assessed as half life incubated for 10 mins measured up to 60 mins in presence of NADPH by LC-MS/MS analysis | Homo sapiens | 11 | microsome format | Scientific Literature | ||
| 5. | ALA5167886 | B | Inhibition of EZH2 (unknown origin) using peptide substrate preincubated for 10 mins followed by substrate addition for 4 hrs by HTRF assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA5167887 | B | Inhibition of MLL1 (unknown origin) using peptide substrate preincubated for 10 mins followed by substrate addition for 4 hrs by HTRF assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 7. | ALA5167888 | B | Inhibition of MLL4 (unknown origin) using peptide substrate preincubated for 10 mins followed by substrate addition for 4 hrs by HTRF assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA5167889 | B | Inhibition of PRMT5 (unknown origin) using histone H4 (1 to 21 residues) peptide/SAM as substrate incubated for 210 mins in presence of SAM by AlphaLISA assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA5167890 | B | Inhibition of NSD2 (unknown origin) using histone H4 (1 to 21 residues) peptide/SAM as substrate incubated for 210 mins in presence of SAM by AlphaLISA assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA5167891 | B | Inhibition of PRMT4 (unknown origin) using histone H4 (1 to 21 residues) peptide/SAM as substrate incubated for 210 mins in presence of SAM by AlphaLISA assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA5167892 | B | Competitive inhibition of PRMT5 (unknown origin) at 0.001 to 100000 nM using histone H4 (1 to 21 residues) as substrate incubated for 120 mins in presence of different concentrations of SAM by AlphaLISA assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA5167893 | B | Competitive inhibition of PRMT5 (unknown origin) at 0.1 to 100 uM using different concentration of histone H4 (1 to 21 residues) as substrate incubated for 120 mins in presence of SAM by AlphaLISA assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA5167894 | B | Competitive inhibition of PRMT5 (unknown origin) in presence of MTA | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA5167895 | F | Antiproliferation activity against human CHL-1 cells assessed as cell growth inhibition incubated for 5 days by CCK-8 assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 15. | ALA5167896 | F | Antiproliferation activity against human SNU-423 cells assessed as cell growth inhibition incubated for 5 days by CCK-8 assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 16. | ALA5167897 | F | Antiproliferation activity against human SNU-449 cells assessed as cell growth inhibition incubated for 5 days by CCK-8 assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA5167898 | F | Antiproliferation activity against human MDA-MB-231 cells assessed as cell growth inhibition incubated for 5 days by CCK-8 assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 18. | ALA5167899 | F | Antiproliferation activity against human MDA-MB-453 cells assessed as cell growth inhibition incubated for 5 days by CCK-8 assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 19. | ALA5167900 | F | Antiproliferation activity against human MV4-11 cells assessed as cell growth inhibition incubated for 5 days by CCK-8 assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 20. | ALA5167901 | F | Antiproliferation activity against human MOLM-13 cells assessed as cell growth inhibition incubated for 5 days by CCK-8 assay | Homo sapiens | 1 | cell-based format | Scientific Literature |
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