| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5138979 | B | Inhibition of PI3Kalpha in rat Rat1 cells assessed as reduction in phosphorylation of AKT at Ser473 residue incubated for 1 hr by cellular assay | Rattus norvegicus | 37 | cell-based format | Scientific Literature | ||
| 2. | ALA5138980 | B | Inhibition of PI3Kbeta in rat Rat1 cells assessed as reduction in phosphorylation of AKT at Ser473 residue incubated for 1 hr by cellular assay | Rattus norvegicus | 37 | cell-based format | Scientific Literature | ||
| 3. | ALA5138981 | B | Inhibition of PI3Kdelta in rat Rat1 cells assessed as reduction in phosphorylation of AKT at Ser473 residue incubated for 1 hr by cellular assay | Rattus norvegicus | 37 | cell-based format | Scientific Literature | ||
| 4. | ALA5138982 | B | Binding affinity to human N-terminal GST-tagged mTOR assessed as phosphorylated 4EBP1 by TR-FRET assay | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 5. | ALA5138983 | B | Binding affinity to tubulin in human A2058 cells assessed as condensed DNA score at 5 uM measured after 6 hrs by DiffQuick staining based microscopic analysis | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 6. | ALA5138984 | B | Binding affinity to tubulin in human A2058 cells assessed as condensed DNA score at 5 uM measured after 24 hrs by DiffQuick staining based microscopic analysis | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 7. | ALA5138988 | A | Brain to blood ratio in OF1 mouse at 1 mg/kg, iv measured at 5 mins post dose by LC-MS/MS analysis | Mus musculus | 11 | organism-based format | Scientific Literature | ||
| 8. | ALA5138989 | A | Brain to blood ratio in OF1 mouse at 1 mg/kg, iv measured at 1 hr post dose by LC-MS/MS analysis | Mus musculus | 11 | organism-based format | Scientific Literature |
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