| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5148363 | B | Displacement of [125-I]-[Sar1Ile8]-angiotensin II from human AT1R expressed in HEK293 cell membrane assessed as inhibition constant by radioligand binding assay | Homo sapiens | 21 | ALA5143706 | cell membrane format | Scientific Literature | |
| 2. | ALA5148364 | B | Displacement of [125-I]-[Sar1Ile8]-angiotensin II from human AT2R expressed in HEK293 cell membrane assessed as inhibition constant by radioligand binding assay | Homo sapiens | 22 | ALA5143706 | cell membrane format | Scientific Literature | |
| 3. | ALA5148365 | A | Metabolic stability in human liver microsomes assessed as half life at 1 uM preincubated for 5 mins followed by NADPH addition and measured upto 60 mins by HPLC-MS/MS analysis | Homo sapiens | 7 | ALA5143706 | microsome format | Scientific Literature | |
| 4. | ALA5148366 | A | Metabolic stability in CD-1 mouse liver microsomes assessed as half life at 1 uM preincubated for 5 mins followed by NADPH addition and measured upto 60 mins by HPLC-MS/MS analysis | Mus musculus | 7 | ALA5143706 | microsome format | Scientific Literature | |
| 5. | ALA5148367 | A | Metabolic stability in Sprague-Dawley rat liver microsomes assessed as half life at 1 uM preincubated for 5 mins followed by NADPH addition and measured upto 60 mins by HPLC-MS/MS analysis | Rattus norvegicus | 7 | ALA5143706 | microsome format | Scientific Literature |
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