| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5142210 | Binding | Inhibition of His-tagged SMARCA4 (unknown origin) (1448 to 1575 residues) using biotinylated ARTKQTARKSTGG-K(Ac)-APR-K(Ac)-QLAT-K(Ac)-AAR-K(Ac)-SAPGG-K as substrate incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | ALA5137085 | single protein format | Scientific Literature | |
| 2. | ALA5142211 | Binding | Inhibition of SMARCA2 (unknown origin) by TR-FRET assay | Homo sapiens | 4 | ALA5137085 | single protein format | Scientific Literature | |
| 3. | ALA5142212 | Binding | Inhibition of PBRM1 bromodomain 5 (unknown origin) by TR-FRET assay | Homo sapiens | 4 | ALA5137085 | single protein format | Scientific Literature | |
| 4. | ALA5142213 | Binding | Inhibition of BRD4 bromodomain 1 (unknown origin) by TR-FRET assay | Homo sapiens | 5 | ALA5137085 | single protein format | Scientific Literature | |
| 5. | ALA5142214 | Binding | Binding affinity to His6/FLAG-tagged SMARCA4 (unknown origin) by isothermal titration calorimetric assay | Homo sapiens | 5 | ALA5137085 | single protein format | Scientific Literature | |
| 6. | ALA5142215 | Binding | Binding affinity to human SMARCA4 (A1448 to S1575 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 5 | ALA5137085 | assay format | Scientific Literature | |
| 7. | ALA5142216 | Binding | Binding affinity to human SMARCA2 (S1337 to Q1486 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 5 | ALA5137085 | assay format | Scientific Literature | |
| 8. | ALA5142217 | Binding | Binding affinity to human PBRM1 bromodomain 5 (S645 to D766 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 5 | ALA5137085 | assay format | Scientific Literature | |
| 9. | ALA5142218 | Binding | Binding affinity to human PBRM1 bromodomain 2 (S178 to E291 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 5 | ALA5137085 | assay format | Scientific Literature | |
| 10. | ALA5142219 | Binding | Inhibition of SMARAC2 isoform B (unknown origin) expressed in U2OS cells co-expressed in NLS-ZsGreen incubated for 1 hrs by cellular target engagement assay | Homo sapiens | 5 | ALA5137085 | cell-based format | Scientific Literature | |
| 11. | ALA5142220 | Binding | Binding affinity to human MHHHHHHGSLVPRGS-tagged SMARAC2 isoform B (S1377 to Q1486 residues) by isothermal titration calorimetric assay | Homo sapiens | 1 | ALA5137085 | cell-based format | Scientific Literature | |
| 12. | ALA5142221 | Binding | Binding affinity to human MHHHHHHGSLVPRGS-tagged SMARAC2 isoform B L1412P/P1413V/S1414N mutant (S1377 to Q1486 residues) by isothermal titration calorimetric assay | Homo sapiens | 1 | ALA5137085 | cell-based format | Scientific Literature | |
| 13. | ALA5142222 | Physicochemical | Kinetic solubility of compound | 2 | ALA5137085 | small-molecule physicochemical format | Scientific Literature | ||
| 14. | ALA5142223 | Physicochemical | Lipophilicity, LogD of compound | 2 | ALA5137085 | small-molecule physicochemical format | Scientific Literature |
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