| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5165189 | A | Metabolic stability of compound in rat liver microsome assessed as half life at 1 uM measured upto 45 mins by LCMS analysis | Rattus norvegicus | 2 | ALA5154875 | microsome format | Scientific Literature | |
| 2. | ALA5165199 | F | Anti-proliferative activity against human MV4-11 cells assessed as inhibition of cell proliferation incubated for 5 days by Cell Titre Glo luminescent assay | Homo sapiens | 40 | ALA5154875 | cell-based format | Scientific Literature | |
| 3. | ALA5165200 | F | Anti-proliferative activity against human K562 cells assessed as inhibition of cell proliferation incubated for 5 days by Cell Titre Glo luminescent assay | Homo sapiens | 40 | ALA5154875 | cell-based format | Scientific Literature | |
| 4. | ALA5165207 | B | Competitive binding affinity to N-terminal 6xHis-SUMO-tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells assessed as inhibition constant using 10-mer-Thr-FAM peptide as substrate incubated for 1 hr by Lantha Screen based TR-FRET assay | Homo sapiens | 39 | ALA5154875 | cell-based format | Scientific Literature | |
| 5. | ALA5165208 | F | Anti-proliferative activity against human MOLM-13 cells assessed as inhibition of cell proliferation incubated for 5 days by Cell Titre Glo luminescent assay | Homo sapiens | 40 | ALA5154875 | cell-based format | Scientific Literature | |
| 6. | ALA5165209 | A | Metabolic stability of compound in rat liver microsome assessed as intrinsic clearance at 1 uM measured upto 45 mins by LCMS analysis | Rattus norvegicus | 2 | ALA5154875 | microsome format | Scientific Literature | |
| 7. | ALA5165210 | F | Selectivity ratio of GI50 for human K562 cells to GI50 for human MV4-11 cells | 40 | ALA5154875 | cell-based format | Scientific Literature |
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