# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA5161714 | B | Inhibition of 20S proteasome subunit beta-5i (unknown origin) using Ac-ANW-AMC as substrate and measured after 30 mins | Homo sapiens | 50 | ALA5154800 | single protein format | Scientific Literature | |
2. | ALA5161715 | B | Inhibition of 20S proteasome subunit beta-5c (unknown origin) using Ac-WLA-AMC as substrate and measured after 30 mins | Homo sapiens | 50 | ALA5154800 | single protein format | Scientific Literature | |
3. | ALA5161716 | B | Selectivity ratio of IC50 for inhibition of 20S proteasome beta 5c subunit (unknown origin) to IC50 for inhibition of 20S proteasome subunit beta-5i | 50 | ALA5154800 | assay format | Scientific Literature | ||
4. | ALA5161717 | F | Antiproliferative activity against human DOHH-2 cells assessed as growth inhibition at 0.2 uM measured after 72 hrs by MTT assay | Homo sapiens | 26 | ALA5154800 | cell-based format | Scientific Literature | |
5. | ALA5161718 | F | Antiproliferative activity against human Pfeiffer cells assessed as growth inhibition at 0.2 uM measured after 72 hrs by MTT assay | Homo sapiens | 26 | ALA5154800 | cell-based format | Scientific Literature | |
6. | ALA5161719 | F | Antiproliferative activity against human HCT-116 cells assessed as growth inhibition at 0.2 uM measured after 72 hrs by MTT assay | Homo sapiens | 26 | ALA5154800 | cell-based format | Scientific Literature | |
7. | ALA5161720 | F | Antiproliferative activity against human HT-29 cells assessed as growth inhibition at 0.2 uM measured after 72 hrs by MTT assay | Homo sapiens | 26 | ALA5154800 | cell-based format | Scientific Literature | |
8. | ALA5161721 | F | Antiproliferative activity against human MCF7 cells assessed as growth inhibition at 0.2 uM measured after 72 hrs by MTT assay | Homo sapiens | 26 | ALA5154800 | cell-based format | Scientific Literature | |
9. | ALA5161723 | F | Antiinflammatory activity against LPS-stimulated human THP-1 cells assessed inhibition of TNF-alpha release at 40 uM measured by ELISA | Homo sapiens | 9 | ALA5154800 | cell-based format | Scientific Literature | |
10. | ALA5161724 | F | Antiinflammatory activity against LPS-stimulated human THP-1 cells assessed inhibition of IL-6 release at 40 uM measured by ELISA | Homo sapiens | 9 | ALA5154800 | cell-based format | Scientific Literature | |
11. | ALA5161725 | B | Inhibition of 20S proteasome subunit beta-1i (unknown origin) using Ac-PAL-AMC as substrate and measured after 30 mins | Homo sapiens | 3 | ALA5154800 | single protein format | Scientific Literature | |
12. | ALA5161726 | B | Inhibition of 20S proteasome subunit beta-1c (unknown origin) using Z-LLE-AMC as substrate and measured after 30 mins | Homo sapiens | 3 | ALA5154800 | single protein format | Scientific Literature | |
13. | ALA5161727 | B | Inhibition of 20S proteasome subunit beta-2i (unknown origin) using Ac-KQL-AMC as substrate and measured after 30 mins | Homo sapiens | 3 | ALA5154800 | single protein format | Scientific Literature | |
14. | ALA5161728 | B | Inhibition of 20S proteasome subunit beta-2c (unknown origin) using Ac-KQL-AMC as substrate and measured after 30 mins | Homo sapiens | 3 | ALA5154800 | single protein format | Scientific Literature |