| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5153031 | B | Inhibition of wild type EGFR (unknown origin) assessed as percent of control activity at 1 uM by radiometric protein kinase-reaction biology assay | Homo sapiens | 27 | ALA5150044 | single protein format | Scientific Literature | |
| 2. | ALA5153032 | B | Inhibition of EGFR (unknown origin) Del19 mutant assessed as percent of control activity at 1 uM by radiometric protein kinase-reaction biology assay | Homo sapiens | 27 | ALA5150044 | single protein format | Scientific Literature | |
| 3. | ALA5153033 | B | Inhibition of EGFR (unknown origin) d747-752/P7535 mutant assessed as percent of control activity at 1 uM by radiometric protein kinase-reaction biology assay | Homo sapiens | 27 | ALA5150044 | single protein format | Scientific Literature | |
| 4. | ALA5153034 | B | Inhibition of wild type EGFR (unknown origin) preincubated with compound 30 mins followed ATP addition incubated for 30 mins by HTRF KinEASE TK assay | Homo sapiens | 27 | ALA5150044 | single protein format | Scientific Literature | |
| 5. | ALA5153035 | B | Inhibition of EGFR (unknown origin) Del19 mutant preincubated with compound 30 mins followed ATP addition incubated for 30 mins by HTRF KinEASE TK assay | Homo sapiens | 27 | ALA5150044 | single protein format | Scientific Literature | |
| 6. | ALA5153036 | B | Inhibition of EGFR (unknown origin) L858R mutant preincubated with compound 30 mins followed ATP addition incubated for 30 mins by HTRF KinEASE TK assay | Homo sapiens | 27 | ALA5150044 | single protein format | Scientific Literature | |
| 7. | ALA5153037 | B | Inhibition of EGFR (unknown origin) L858R/T790M mutant preincubated with compound 30 mins followed ATP addition incubated for 30 mins by HTRF KinEASE TK assay | Homo sapiens | 27 | ALA5150044 | single protein format | Scientific Literature | |
| 8. | ALA5153044 | B | Inhibition of EGER d746-750 mutant (unknown origin) assessed as percent of control activity at 1 uM by radiometric protein kinase-reaction biology assay | Homo sapiens | 1 | ALA5150044 | single protein format | Scientific Literature | |
| 9. | ALA5153045 | B | Inhibition of FLT3 D835V mutant (unknown origin) assessed as percent of control activity at 1 uM by radiometric protein kinase-reaction biology assay | Homo sapiens | 1 | ALA5150044 | single protein format | Scientific Literature | |
| 10. | ALA5153046 | B | Inhibition of EGFR d747-751/Sins mutant (unknown origin) assessed as percent of control activity at 1 uM by radiometric protein kinase-reaction biology assay | Homo sapiens | 1 | ALA5150044 | single protein format | Scientific Literature | |
| 11. | ALA5153047 | B | Inhibition of EGFR d747-752/P7535 mutant (unknown origin) assessed as percent of control activity at 1 uM by radiometric protein kinase-reaction biology assay | Homo sapiens | 1 | ALA5150044 | single protein format | Scientific Literature | |
| 12. | ALA5153048 | B | Inhibition of EGFR L858R mutant (unknown origin) assessed as percent of control activity at 1 uM by radiometric protein kinase-reaction biology assay | Homo sapiens | 1 | ALA5150044 | single protein format | Scientific Literature | |
| 13. | ALA5153049 | B | Inhibition of EGFR d752-759 mutant (unknown origin) assessed as percent of control activity at 1 uM by radiometric protein kinase-reaction biology assay | Homo sapiens | 1 | ALA5150044 | single protein format | Scientific Literature | |
| 14. | ALA5153050 | B | Inhibition of EGFR G719S mutant (unknown origin) assessed as percent of control activity at 1 uM by radiometric protein kinase-reaction biology assay | Homo sapiens | 1 | ALA5150044 | single protein format | Scientific Literature | |
| 15. | ALA5153051 | B | Inhibition of FLT3 D835Y mutant (unknown origin) assessed as percent of control activity at 1 uM by radiometric protein kinase-reaction biology assay | Homo sapiens | 1 | ALA5150044 | single protein format | Scientific Literature | |
| 16. | ALA5153052 | B | Inhibition of EGFR L8610 mutant (unknown origin) assessed as percent of control activity at 1 uM by radiometric protein kinase-reaction biology assay | Homo sapiens | 1 | ALA5150044 | assay format | Scientific Literature | |
| 17. | ALA5153053 | B | Inhibition of EGFR G719C mutant (unknown origin) assessed as percent of control activity at 1 uM by radiometric protein kinase-reaction biology assay | Homo sapiens | 1 | ALA5150044 | single protein format | Scientific Literature | |
| 18. | ALA5153054 | B | Inhibition of FLT3 ITD/D835V mutant (unknown origin) assessed as percent of control activity at 1 uM by radiometric protein kinase-reaction biology assay | Homo sapiens | 1 | ALA5150044 | single protein format | Scientific Literature | |
| 19. | ALA5153056 | F | Antiproliferative activity against mouse BaF3 cells expressing L858R assessed as cell viability measured after 72 hrs hrs by CellTiter Glo assay | Mus musculus | 9 | ALA5150044 | cell-based format | Scientific Literature | |
| 20. | ALA5153057 | F | Antiproliferative activity against mouse BaF3 cells expressing L858R/C797S assessed as cell viability measured after 72 hrs hrs by CellTiter Glo assay | Mus musculus | 8 | ALA5150044 | cell-based format | Scientific Literature |
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