# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA5134825 | Binding | Inhibition of PKN2 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysis | Homo sapiens | 15 | ALA5131476 | single protein format | Scientific Literature | |
2. | ALA5134826 | Binding | Inhibition of PKN2 (unknown origin) by TR-FRET-based tracer displacement assay | Homo sapiens | 15 | ALA5131476 | single protein format | Scientific Literature | |
3. | ALA5134827 | Binding | Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysis | Homo sapiens | 15 | ALA5131476 | single protein format | Scientific Literature | |
4. | ALA5134828 | Binding | Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay | Homo sapiens | 15 | ALA5131476 | single protein format | Scientific Literature | |
5. | ALA5134829 | Binding | Selectivity index, ratio of IC50 for inhibition of PKN1 (unknown origin) to IC50 for inhibition of PKN2 (unknown origin) | Homo sapiens | 15 | ALA5131476 | assay format | Scientific Literature | |
6. | ALA5134833 | Binding | Inhibition of NanoLuc-PKN2 (ser646-cys984)(unknown origin) expressed in HEK293 cells by cell-based NanoBRET target engagement assay | Homo sapiens | 4 | ALA5131476 | cell-based format | Scientific Literature | |
7. | ALA5134835 | Toxicity | Toxicity in human HeLa cells assessed as cell viability at 50 uM incubated for 24 hrs by MTT assay | Homo sapiens | 3 | ALA5131476 | cell-based format | Scientific Literature |