| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5131264 | T | Displacement of [3H]-HS665 from MOR in rat brain membranes | Rattus norvegicus | 15 | cell membrane format | Scientific Literature | ||
| 2. | ALA5131265 | T | Displacement of [3H]-HS665 from DOR in rat brain membranes | Rattus norvegicus | 15 | cell membrane format | Scientific Literature | ||
| 3. | ALA5131266 | B | Displacement of [3H]-HS665 from KOR in guinea pig brain membranes | Cavia porcellus | 15 | cell membrane format | Scientific Literature | ||
| 4. | ALA5131267 | F | Agonist activity at KOR in guinea pig brain membranes assessed as stimulation of [35S]GTPgammaS binding measured after 1 hr by liquid scintillation counting analysis relative to control | Cavia porcellus | 15 | cell membrane format | Scientific Literature | ||
| 5. | ALA5131268 | F | Agonist activity at KOR in guinea pig brain membranes assessed as stimulation of [35S]GTPgammaS binding measured after 1 hr by liquid scintillation counting analysis | Cavia porcellus | 15 | cell membrane format | Scientific Literature | ||
| 6. | ALA5131269 | F | Antinociceptive activity in CD-1 mouse assessed as maximum possible effect at 10 nmol, icv measured after 15 to 120 mins by tail-flick test | Mus musculus | 6 | organism-based format | Scientific Literature | ||
| 7. | ALA5131273 | A | Cmax in C57/BL6 mouse plasma at 13.9 mg/kg, iv administered via bolus by LC-MS/MS analysis | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 8. | ALA5131274 | A | Tmax in C57/BL6 mouse plasma at 13.9 mg/kg, iv administered via bolus by LC-MS/MS analysis | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 9. | ALA5131275 | A | Half life in C57/BL6 mouse plasma at 13.9 mg/kg, iv administered via bolus by LC-MS/MS analysis | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 10. | ALA5131276 | A | AUC (infinity) in C57/BL6 mouse plasma at 13.9 mg/kg, iv administered via bolus by LC-MS/MS analysis | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 11. | ALA5131277 | A | Drug uptake in C57/BL6 mouse brain at 13.9 mg/kg, iv administered via bolus by LC-MS/MS analysis | Mus musculus | 2 | organism-based format | Scientific Literature |
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