| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5149637 | B | Inhibition of full-length N-terminal His-TEV-tagged inactive form of MSK1 (2 to 802 residues) (unknown origin) expressed in HEK293 cells using FAM-PSKPAATRKRRWSAPESR-NH2 as substrate preincubated for 1 hr followed by activation with ERK2 and substrate addition measured after 2 hrs by microfluidic chip based electrophoresis | Homo sapiens | 27 | ALA5143742 | cell-based format | Scientific Literature | |
| 2. | ALA5149640 | B | Inhibition of MSK2 (unknown origin) FAM-PSKPAATRKRRWSAPESR-NH2 as substrate preincubated for 1 hr followed by activation with ERK2 and substrate addition measured after 2 hrs by microfluidic chip based electrophoresis | Homo sapiens | 5 | ALA5143742 | cell-based format | Scientific Literature | |
| 3. | ALA5149677 | P | Glutathione reactivity in pH 7.4 phosphate buffered assessed as GSH-adduct formation at 10 uM measured after 30 mins by UPLC-QTOF analysis | 5 | ALA5143742 | small-molecule physicochemical format | Scientific Literature | ||
| 4. | ALA5149678 | A | Glutathione reactivity in human liver microsomes assessed as GSH-adduct formation at 10 uM measured after 30 mins by UPLC-QTOF analysis | Homo sapiens | 5 | ALA5143742 | microsome format | Scientific Literature | |
| 5. | ALA5149679 | B | Inhibition of RSK1 (unknown origin) up to 10 uM | Homo sapiens | 2 | ALA5143742 | single protein format | Scientific Literature | |
| 6. | ALA5149680 | B | Inhibition of RSK2 (unknown origin) up to 10 uM | Homo sapiens | 2 | ALA5143742 | single protein format | Scientific Literature | |
| 7. | ALA5149681 | B | Inhibition of PLK3 (unknown origin) up to 10 uM | Homo sapiens | 2 | ALA5143742 | single protein format | Scientific Literature |
The page will load shortly, Thanks for your patience!