| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5117929 | B | Inhibition of EGFR del18/T790M/C797S triple mutant (unknown origin) using TK as substrate incubated for 120 mins in the presence of ATP by HTRF assay | Homo sapiens | 20 | single protein format | Scientific Literature | ||
| 2. | ALA5117930 | B | Inhibition of EGFR L858R/T790M/C797S triple mutant (unknown origin) using TK as substrate incubated for 120 mins in the presence of ATP by HTRF assay | Homo sapiens | 21 | single protein format | Scientific Literature | ||
| 3. | ALA5117932 | F | Antiproliferative activity against mouse BaF3 cells harboring del18/T790M/C797S triple mutant assessed as cell growth inhibition incubated for 72 hrs by cell titre glo luminescence assay | Mus musculus | 21 | cell-based format | Scientific Literature | ||
| 4. | ALA5117934 | A | Cmax in mouse at 5 mg/kg measured upto 24 hrs by LC-MS/MS analysis | Mus musculus | 7 | organism-based format | Scientific Literature | ||
| 5. | ALA5117935 | A | AUC(0 to t) in mouse at 5 mg/kg measured upto 24 hrs by LC-MS/MS analysis | Mus musculus | 7 | organism-based format | Scientific Literature | ||
| 6. | ALA5117936 | A | AUC(0 to infinity) in mouse at 5 mg/kg measured upto 24 hrs by LC-MS/MS analysis | Mus musculus | 7 | organism-based format | Scientific Literature | ||
| 7. | ALA5117937 | A | Half-life in mouse at 5 mg/kg measured upto 24 hrs by LC-MS/MS analysis | Mus musculus | 7 | organism-based format | Scientific Literature | ||
| 8. | ALA5117938 | A | MRT in mouse at 5 mg/kg measured upto 24 hrs by LC-MS/MS analysis | Mus musculus | 6 | organism-based format | Scientific Literature | ||
| 9. | ALA5117939 | B | Inhibition of ABL (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 10. | ALA5117940 | B | Inhibition of MET (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA5117941 | B | Inhibition of RET (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA5117942 | B | Inhibition of AURA (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA5117943 | B | Inhibition of AXL (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA5117944 | B | Inhibition of EphA1 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA5117945 | B | Inhibition of EphB2 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA5117946 | B | Inhibition of FER (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA5117947 | B | Inhibition of PDGFRbeta (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA5117948 | B | Inhibition of ROS (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA5117949 | B | Inhibition of JAK2 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 20. | ALA5117950 | B | Inhibition of P38alpha (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature |
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