# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA5115996 | F | Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP level | Homo sapiens | 43 | ALA5113417 | cell-based format | Scientific Literature | |
2. | ALA5115997 | A | Metabolic stability in human liver microsomes assessed as intrinsic clearance | Homo sapiens | 2 | ALA5113417 | microsome format | Scientific Literature | |
3. | ALA5115998 | A | Metabolic stability in rat liver microsomes assessed as intrinsic clearance | Rattus norvegicus | 2 | ALA5113417 | microsome format | Scientific Literature | |
4. | ALA5116002 | A | Cmax in Sprague-Dawley rat at 10 mg/kg, po | Rattus norvegicus | 2 | ALA5113417 | organism-based format | Scientific Literature | |
5. | ALA5116003 | A | AUC(0 to infinity) in Sprague-Dawley rat at 10 mg/kg, po | Rattus norvegicus | 2 | ALA5113417 | organism-based format | Scientific Literature | |
6. | ALA5116004 | A | Oral bioavailability in Sprague-Dawley rat at 10 mg/kg | Rattus norvegicus | 2 | ALA5113417 | organism-based format | Scientific Literature | |
7. | ALA5116005 | F | Agonist activity at human SST1 | Homo sapiens | 2 | ALA5113417 | assay format | Scientific Literature | |
8. | ALA5116006 | F | Agonist activity at human SST2 | Homo sapiens | 3 | ALA5113417 | assay format | Scientific Literature | |
9. | ALA5116007 | F | Agonist activity at human SST3 | Homo sapiens | 2 | ALA5113417 | assay format | Scientific Literature | |
10. | ALA5116008 | F | Agonist activity at human SST4 | Homo sapiens | 2 | ALA5113417 | assay format | Scientific Literature | |
11. | ALA5116009 | F | Agonist activity at rat SST5 | Rattus norvegicus | 2 | ALA5113417 | assay format | Scientific Literature | |
12. | ALA5116012 | T | Inhibition of hERG by patch clamp assay | Homo sapiens | 2 | ALA5113417 | assay format | Scientific Literature | |
13. | ALA5116013 | A | Inhibition of CYP2C9 (unknown origin) by fluorescent assay | Homo sapiens | 1 | ALA5113417 | single protein format | Scientific Literature | |
14. | ALA5116014 | A | Inhibition of CYP2C19 (unknown origin) by fluorescent assay | Homo sapiens | 1 | ALA5113417 | single protein format | Scientific Literature | |
15. | ALA5116015 | A | Inhibition of CYP2D6 (unknown origin) | Homo sapiens | 2 | ALA5113417 | single protein format | Scientific Literature | |
16. | ALA5116016 | A | Inhibition of CYP2D6 (unknown origin) preincubated for 30 mins | Homo sapiens | 2 | ALA5113417 | single protein format | Scientific Literature | |
17. | ALA5116017 | A | Inhibition of CYP3A4 (unknown origin) | Homo sapiens | 2 | ALA5113417 | single protein format | Scientific Literature | |
18. | ALA5116018 | A | Inhibition of CYP3A4 (unknown origin) preincubated for 30 mins | Homo sapiens | 2 | ALA5113417 | single protein format | Scientific Literature | |
19. | ALA5116019 | A | Metabolic stability in human liver microsomes assessed as half life | Homo sapiens | 1 | ALA5113417 | microsome format | Scientific Literature | |
20. | ALA5116020 | A | Metabolic stability in rat liver microsomes assessed as half life | Rattus norvegicus | 1 | ALA5113417 | microsome format | Scientific Literature |