# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA5128931 | Binding | Inhibition of full length C-terminal His-tagged HDAC3 (unknown origin)/N-terminal GST-tagged NCoR2 (unknown origin) assessed as inhibition constant (Ki) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate measured every 30 sec for 60 mins by fluorescence based assay | Homo sapiens | 3 | ALA5126568 | protein complex format | Scientific Literature | |
2. | ALA5128932 | Binding | Inhibition of full length C-terminal FLAG-tagged HDAC2 (unknown origin) assessed as inhibition constant (Ki) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate measured every 30 sec for 60 mins by fluorescence based assay | Homo sapiens | 3 | ALA5126568 | single protein format | Scientific Literature | |
3. | ALA5128933 | Binding | Inhibition of full length C-terminal His-tagged HDAC1 (unknown origin) assessed as inhibition constant (Ki) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate measured every 30 sec for 60 mins by fluorescence based assay | Homo sapiens | 3 | ALA5126568 | single protein format | Scientific Literature | |
4. | ALA5128934 | Binding | Inhibition of full length C-terminal His-tagged HDAC3 (unknown origin)/N-terminal GST-tagged NCoR2 (unknown origin) assessed as equilibrium inhibition constant (Ki,1) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate measured every 30 sec for 60 mins by fluorescence based assay | Homo sapiens | 3 | ALA5126568 | protein complex format | Scientific Literature | |
5. | ALA5128935 | Binding | Inhibition of full length C-terminal FLAG-tagged HDAC2 (unknown origin) assessed as equilibrium inhibition constant (Ki,1) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate measured every 30 sec for 60 mins by fluorescence based assay | Homo sapiens | 2 | ALA5126568 | single protein format | Scientific Literature | |
6. | ALA5128936 | Binding | Inhibition of full length C-terminal His-tagged HDAC1 (unknown origin) assessed as equilibrium inhibition constant (Ki,1) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate measured every 30 sec for 60 mins by fluorescence based assay | Homo sapiens | 2 | ALA5126568 | single protein format | Scientific Literature | |
7. | ALA5128937 | Binding | Inhibition of full length C-terminal His-tagged HDAC3 (unknown origin)/N-terminal GST-tagged NCoR2 (unknown origin) assessed as rate constant (k-2) of EI complex using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate measured every 30 sec for 60 mins by fluorescence based assay | Homo sapiens | 3 | ALA5126568 | protein complex format | Scientific Literature | |
8. | ALA5128938 | Binding | Inhibition of full length C-terminal FLAG-tagged HDAC2 (unknown origin) assessed as rate constant (k-2) of EI complex using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate measured every 30 sec for 60 mins by fluorescence based assay | Homo sapiens | 2 | ALA5126568 | single protein format | Scientific Literature | |
9. | ALA5128939 | Binding | Inhibition of full length C-terminal His-tagged HDAC1 (unknown origin) assessed as rate constant (k-2) of EI complex using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate measured every 30 sec for 60 mins by fluorescence based assay | Homo sapiens | 2 | ALA5126568 | single protein format | Scientific Literature | |
10. | ALA5128940 | Binding | Inhibition of full length C-terminal His-tagged HDAC3 (unknown origin)/N-terminal GST-tagged NCoR2 (unknown origin) assessed as rate constant (k2) of EI complex using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate measured every 30 sec for 60 mins by fluorescence based assay | Homo sapiens | 3 | ALA5126568 | protein complex format | Scientific Literature | |
11. | ALA5128941 | Binding | Inhibition of full length C-terminal FLAG-tagged HDAC2 (unknown origin) assessed as rate constant (k2) of EI complex using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate measured every 30 sec for 60 mins by fluorescence based assay | Homo sapiens | 2 | ALA5126568 | single protein format | Scientific Literature | |
12. | ALA5128942 | Binding | Inhibition of full length C-terminal His-tagged HDAC1 (unknown origin) assessed as rate constant (k2) of EI complex using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate measured every 30 sec for 60 mins by fluorescence based assay | Homo sapiens | 2 | ALA5126568 | single protein format | Scientific Literature | |
13. | ALA5128945 | Binding | Inhibition of full length C-terminal His-tagged HDAC1 (unknown origin) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate incubated for 30 mins by fluorescence based assay | Homo sapiens | 2 | ALA5126568 | single protein format | Scientific Literature | |
14. | ALA5128946 | Binding | Inhibition of full length C-terminal His-tagged HDAC1 (unknown origin) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured after 30 mins by fluorescence based assay | Homo sapiens | 2 | ALA5126568 | single protein format | Scientific Literature | |
15. | ALA5128947 | Binding | Inhibition of full length C-terminal His-tagged HDAC1 (unknown origin) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate preincubated with enzyme for 1 hrs followed by substrate addition and measured after 30 mins by fluorescence based assay | Homo sapiens | 2 | ALA5126568 | single protein format | Scientific Literature | |
16. | ALA5128948 | Binding | Inhibition of full length C-terminal His-tagged HDAC1 (unknown origin) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate preincubated with enzyme for 2 hrs followed by substrate addition and measured after 30 mins by fluorescence based assay | Homo sapiens | 2 | ALA5126568 | single protein format | Scientific Literature | |
17. | ALA5128949 | Binding | Inhibition of full length C-terminal FLAG-tagged HDAC2 (unknown origin) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate incubated for 30 mins by fluorescence based assay | Homo sapiens | 2 | ALA5126568 | single protein format | Scientific Literature | |
18. | ALA5128950 | Binding | Inhibition of full length C-terminal FLAG-tagged HDAC2 (unknown origin) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured after 30 mins by fluorescence based assay | Homo sapiens | 2 | ALA5126568 | single protein format | Scientific Literature | |
19. | ALA5128951 | Binding | Inhibition of full length C-terminal FLAG-tagged HDAC2 (unknown origin) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate preincubated with enzyme for 1 hrs followed by substrate addition and measured after 30 mins by fluorescence based assay | Homo sapiens | 2 | ALA5126568 | single protein format | Scientific Literature | |
20. | ALA5128952 | Binding | Inhibition of full length C-terminal FLAG-tagged HDAC2 (unknown origin) using (Ac-Leu-Gly-Lys(Ac)-AMC as substrate preincubated with enzyme for 2 hrs followed by substrate addition and measured after 30 mins by fluorescence based assay | Homo sapiens | 2 | ALA5126568 | single protein format | Scientific Literature |