| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5106511 | F | Antiinflammatory activity against mouse air pouch model of carrageenan-induced oedema assessed as reduction in total inflammatory cell volume into air pouch at 0.6 to 6 mg/kg, po administered as single dose for 1 hr followed byb carrageenan administration | Mus musculus | 1 | ALA5104173 | organism-based format | Scientific Literature | |
| 2. | ALA5106512 | B | Inhibition of recombinant human SSAO | Homo sapiens | 10 | ALA5104173 | single protein format | Scientific Literature | |
| 3. | ALA5106513 | B | Inhibition of human recombinant MAO-B | Homo sapiens | 10 | ALA5104173 | single protein format | Scientific Literature | |
| 4. | ALA5106514 | B | Inhibition of human recombinant MAO-A | Homo sapiens | 10 | ALA5104173 | single protein format | Scientific Literature | |
| 5. | ALA5106515 | B | Inhibition of human recombinant DAO | Homo sapiens | 10 | ALA5104173 | single protein format | Scientific Literature | |
| 6. | ALA5106516 | B | Selectivity index, ratio of IC50 for inhibition of human recombinant MAO-A to IC50 for inhibition of recombinant human SSAO | Homo sapiens | 5 | ALA5104173 | assay format | Scientific Literature | |
| 7. | ALA5106517 | B | Selectivity index, ratio of IC50 for inhibition of human recombinant MAO-A to IC50 for inhibition of recombinant human MAO-B | Homo sapiens | 5 | ALA5104173 | assay format | Scientific Literature | |
| 8. | ALA5106518 | B | Inhibition of SSAO in HMEC cells | Homo sapiens | 1 | ALA5104173 | cell-based format | Scientific Literature | |
| 9. | ALA5106519 | B | Inhibition of rat SSAO | Rattus norvegicus | 1 | ALA5104173 | single protein format | Scientific Literature | |
| 10. | ALA5106520 | B | Inhibition of mouse muscle MAO-B | Mus musculus | 1 | ALA5104173 | tissue-based format | Scientific Literature | |
| 11. | ALA5106521 | B | Inhibition of recombinant human LOXL-2 | Homo sapiens | 1 | ALA5104173 | single protein format | Scientific Literature | |
| 12. | ALA5106522 | B | Inhibition of bovine aorta LOX | Bos taurus | 1 | ALA5104173 | tissue-based format | Scientific Literature | |
| 13. | ALA5106523 | B | Inhibition of LSD1 (unknown origin) | Homo sapiens | 1 | ALA5104173 | single protein format | Scientific Literature | |
| 14. | ALA5106524 | A | Plasma protein binding in human | Homo sapiens | 1 | ALA5104173 | cell-free format | Scientific Literature | |
| 15. | ALA5106525 | A | Plasma protein binding in rat | Rattus norvegicus | 1 | ALA5104173 | cell-free format | Scientific Literature | |
| 16. | ALA5106526 | A | Plasma protein binding in dog | Canis lupus familiaris | 1 | ALA5104173 | cell-free format | Scientific Literature | |
| 17. | ALA5106527 | A | Stability in human microsomes measured after 1 hr | Homo sapiens | 1 | ALA5104173 | microsome format | Scientific Literature | |
| 18. | ALA5106528 | A | Stability in rat microsomes measured after 1 hr | Rattus norvegicus | 1 | ALA5104173 | microsome format | Scientific Literature | |
| 19. | ALA5106529 | A | Stability in dog microsomes measured after 1 hr | Canis lupus familiaris | 1 | ALA5104173 | microsome format | Scientific Literature | |
| 20. | ALA5106530 | A | Stability in human hepatocytes assessed as parent compound remaining measured after 1 hr | Homo sapiens | 1 | ALA5104173 | cell-based format | Scientific Literature |
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