| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5163713 | B | Inhibition of TRIM24 (unknown origin) at 20 uM measured alphascreen assay relative to control | Homo sapiens | 39 | ALA5154837 | single protein format | Scientific Literature | |
| 2. | ALA5163714 | B | Inhibition of TRIM24 (unknown origin) measured alphascreen assay | Homo sapiens | 39 | ALA5154837 | single protein format | Scientific Literature | |
| 3. | ALA5163715 | B | Inhibition of BRPF1 (unknown origin) measured alphascreen assay | Homo sapiens | 1 | ALA5154837 | single protein format | Scientific Literature | |
| 4. | ALA5163716 | F | Antiproliferative activity against human LNCaP C4-2B cells measured after 96 hrs by Cell Titer-Glo assay | Homo sapiens | 2 | ALA5154837 | cell-based format | Scientific Literature | |
| 5. | ALA5163717 | F | Antiproliferative activity against human LNCaP cells measured after 96 hrs by Cell Titer-Glo assay | Homo sapiens | 2 | ALA5154837 | cell-based format | Scientific Literature | |
| 6. | ALA5163718 | F | Antiproliferative activity against human 22Rv1 cells measured after 96 hrs by Cell Titer-Glo assay | Homo sapiens | 2 | ALA5154837 | cell-based format | Scientific Literature | |
| 7. | ALA5163719 | F | Inhibition of clonogenicity in human LNCaP C4-2B cells assessed as reduction in colony formation at 1 uM measured by crystal violet staining based analysis | Homo sapiens | 1 | ALA5154837 | cell-based format | Scientific Literature | |
| 8. | ALA5163720 | F | Inhibition of clonogenicity in human 22Rv1 cells assessed as reduction in colony formation at 1 uM measured by crystal violet staining based analysis | Homo sapiens | 1 | ALA5154837 | cell-based format | Scientific Literature | |
| 9. | ALA5163721 | F | Downregulation of full-length AR mRNA expression in human 22Rv1 cells at 5 uM measured by RT-PCR analysis | Homo sapiens | 1 | ALA5154837 | cell-based format | Scientific Literature | |
| 10. | ALA5163722 | F | Downregulation of AR-V7 mRNA expression in human 22Rv1 cells at 5 uM measured by RT-PCR analysis | Homo sapiens | 1 | ALA5154837 | cell-based format | Scientific Literature | |
| 11. | ALA5163723 | F | Downregulation of PSA mRNA expression in human 22Rv1 cells at 5 uM measured by RT-PCR analysis | Homo sapiens | 1 | ALA5154837 | cell-based format | Scientific Literature | |
| 12. | ALA5163724 | F | Downregulation of KLK2 mRNA expression in human 22Rv1 cells at 5 uM measured by RT-PCR analysis | Homo sapiens | 1 | ALA5154837 | cell-based format | Scientific Literature | |
| 13. | ALA5163725 | F | Downregulation of TMPRSS2 mRNA expression in human 22Rv1 cells at 5 uM measured by RT-PCR analysis | Homo sapiens | 1 | ALA5154837 | cell-based format | Scientific Literature | |
| 14. | ALA5163726 | F | Downregulation of C-MYC mRNA expression in human 22Rv1 cells at 5 uM measured by RT-PCR analysis | Homo sapiens | 1 | ALA5154837 | cell-based format | Scientific Literature | |
| 15. | ALA5163727 | F | Suppression of PSA gene expression in human LNCaP cells assessed as mRNA level at 0.4 to 10 uM measured by luciferase gene reporter assay | Homo sapiens | 1 | ALA5154837 | cell-based format | Scientific Literature | |
| 16. | ALA5163728 | A | Apparent permeability of the compound across apical to basolateral side in human Caco-2 cells at 10 uM incubated for 120 mins and measured by LC-MS/MS analysis | Homo sapiens | 4 | ALA5154837 | cell-based format | Scientific Literature | |
| 17. | ALA5163729 | A | Apparent permeability of the compound across basolateral to apical side in human Caco-2 cells at 10 uM incubated for 120 mins and measured by LC-MS/MS analysis | Homo sapiens | 4 | ALA5154837 | cell-based format | Scientific Literature | |
| 18. | ALA5163730 | A | Efflux ratio of apparent permeability from basolateral to apical side over apical to basolateral side in human Caco-2 cells at 10 uM incubated for 120 mins and measured by LC-MS/MS analysis | Homo sapiens | 2 | ALA5154837 | cell-based format | Scientific Literature | |
| 19. | ALA5163731 | A | Apparent permeability of the compound across apical to basolateral side in human Caco-2 cells at 10 uM incubated for 120 mins assessed as drug recovery and measured by LC-MS/MS analysis | Homo sapiens | 4 | ALA5154837 | cell-based format | Scientific Literature | |
| 20. | ALA5163732 | A | Apparent permeability of the compound across basolateral to apical side in human Caco-2 cells at 10 uM incubated for 120 mins assessed as drug recovery and measured by LC-MS/MS analysis | Homo sapiens | 4 | ALA5154837 | cell-based format | Scientific Literature |
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