# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA5153779 | B | Inhibition of full-length USP7 (unknown origin) using ubiquitin-rhodamine 110 as substrate preincubated for 30 mins followed by substrate addition and measured after 2 hrs by microplate spectrophotometer analysis | Homo sapiens | 40 | single protein format | Scientific Literature | ||
2. | ALA5153780 | B | Inhibition of USP2 (unknown origin) at 10 uM using ubiquitin-rhodamine 110 as substrate preincubated for 30 mins followed by substrate addition and measured after 2 hrs by microplate spectrophotometer analysis | Homo sapiens | 6 | single protein format | Scientific Literature | ||
3. | ALA5153781 | B | Inhibition of USP9x (unknown origin) at 10 uM using ubiquitin-rhodamine 110 as substrate preincubated for 30 mins followed by substrate addition and measured after 2 hrs by microplate spectrophotometer analysis | Homo sapiens | 6 | single protein format | Scientific Literature | ||
4. | ALA5153782 | B | Inhibition of USP11 (unknown origin) at 10 uM using ubiquitin-rhodamine 110 as substrate preincubated for 30 mins followed by substrate addition and measured after 2 hrs by microplate spectrophotometer analysis | Homo sapiens | 6 | single protein format | Scientific Literature | ||
5. | ALA5153783 | B | Inhibition of USP25 (unknown origin) at 10 uM using ubiquitin-rhodamine 110 as substrate preincubated for 30 mins followed by substrate addition and measured after 2 hrs by microplate spectrophotometer analysis | Homo sapiens | 6 | single protein format | Scientific Literature | ||
6. | ALA5153784 | B | Inhibition of USP28 (unknown origin) at 10 uM using ubiquitin-rhodamine 110 as substrate preincubated for 30 mins followed by substrate addition and measured after 2 hrs by microplate spectrophotometer analysis | Homo sapiens | 6 | single protein format | Scientific Literature | ||
7. | ALA5153785 | B | Inhibition of USP47 (unknown origin) at 10 uM using ubiquitin-rhodamine 110 as substrate preincubated for 30 mins followed by substrate addition and measured after 2 hrs by microplate spectrophotometer analysis | Homo sapiens | 6 | single protein format | Scientific Literature | ||
8. | ALA5153786 | B | Inhibition of UCH-L1 (unknown origin) at 10 uM using ubiquitin-rhodamine 110 as substrate preincubated for 30 mins followed by substrate addition and measured after 2 hrs by microplate spectrophotometer analysis | Homo sapiens | 6 | single protein format | Scientific Literature | ||
9. | ALA5153787 | B | Inhibition of UCH-L5 (unknown origin) at 10 uM using ubiquitin-rhodamine 110 as substrate preincubated for 30 mins followed by substrate addition and measured after 2 hrs by microplate spectrophotometer analysis | Homo sapiens | 6 | single protein format | Scientific Literature | ||
10. | ALA5153788 | B | Inhibition of USP11 (unknown origin) at 40 uM using ubiquitin-rhodamine 110 as substrate preincubated for 30 mins followed by substrate addition and measured after 2 hrs by microplate spectrophotometer analysis relative to control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
11. | ALA5153789 | B | Inhibition of USP47 (unknown origin) at 40 uM using ubiquitin-rhodamine 110 as substrate preincubated for 30 mins followed by substrate addition and measured after 2 hrs by microplate spectrophotometer analysis relative to control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
12. | ALA5153790 | B | Binding affinity to human USP7 (208 to 560 residues) by SPR method | Homo sapiens | 8 | single protein format | Scientific Literature | ||
13. | ALA5153791 | A | Metabolic stability in rat liver microsomes assessed as half life | Rattus norvegicus | 14 | microsome format | Scientific Literature | ||
14. | ALA5153792 | A | Apparent permeability across apical to basolateral side in human Caco-2 cells | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
15. | ALA5153793 | A | Apparent permeability across basolateral to apical side in human Caco-2 cells | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
16. | ALA5153794 | A | Efflux ratio of apparent permeability across basolateral to apical side over apical to basolateral side in human Caco2 cells | Homo sapiens | 12 | cell-based format | Scientific Literature |