| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5158072 | B | Inhibition of human recombinant NEK1 (1 to 505 residues) using RLGRDKYKTLRQIRQ as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric scintillation counting assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 2. | ALA5158073 | B | Inhibition of human recombinant NEK1 (1 to 505 residues) assessed as residual activity at 1 uM using RLGRDKYKTLRQIRQ as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by radiometric scintillation counting assay relative to control | Homo sapiens | 19 | single protein format | Scientific Literature | ||
| 3. | ALA5158074 | B | Inhibition of human recombinant NEK1 (1 to 505 residues) using ULight-p70 S6K peptide as substrate incubated for 30 mins by LANCE Ultra TR-FRET assay | Homo sapiens | 19 | single protein format | Scientific Literature | ||
| 4. | ALA5158076 | B | Inhibition of recombinant human full length IKKbeta assessed as residual activity at 1 uM using peptide as substrate incubated for 40 mins in presence of [gamma 33P]-ATP by radiometric scintillation counting assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 5. | ALA5158077 | B | Inhibition of human full length recombinant IKKalpha assessed as residual activity at 1 uM using peptide as substrate incubated for 40 mins in presence of [gamma 33P]-ATP by radiometric scintillation counting assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA5158078 | B | Inhibition of human full length recombinant TLK1 assessed as residual activity at 1 uM using casein as substrate incubated for 40 mins in presence of [gamma 33P]-ATP by radiometric scintillation counting assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 7. | ALA5158079 | B | Inhibition of human full length recombinant NEK11 assessed as residual activity at 1 uM using myelin basic protein as substrate incubated for 40 mins in presence of [gamma 33P]-ATP by radiometric scintillation counting assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA5158080 | B | Inhibition of human recombinant ABL (27 to end residues) assessed as residual activity at 1 uM using EAIYAAPFAKKK as substrate incubated for 40 mins in presence of [gamma33P-ATP] by radiometric scintillation counting analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA5158081 | B | Inhibition of human GSK3beta (2 to end residues) assessed as residual activity using YRRAAVPPSPSLSRHSSPHQS(p) EDEEE as substrate at 1 uM incubated for 40 mins in presence of [gamma 33P]-ATP by radiometric scintillation counting assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA5158082 | B | Inhibition of recombinant human full length SAPK2a assessed as residual activity at 1 uM using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting method relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA5158083 | B | Inhibition of recombinant human Lyn assessed as residual activity at 1 uM using poly(Glu, Tyr) 4:1 as substrate after 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA5158084 | B | Inhibition of recombinant human EphB4 (561 to end residues) assessed as residual activity at 1 uM using poly(Glu, Tyr) 4:1 as substrate at 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA5158085 | B | Inhibition of human full length recombinant CDK1/CyclinB assessed as residual activity at 1 uM using histone H1 as substrate incubated for 40 mins in in presence of [gamma 33P]-ATP by radiometric scintillation counting assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA5158086 | B | Inhibition of recombinant full length human BRK assessed as residual activity at 1 uM using poly(Glu, Tyr) 4:1 as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA5158087 | B | Inhibition of human c-Raf (Raf-1) Y340D/Y341D mutant (306 to end) as residual activity at 1 uM using inactive MEK1 as substrate incubated for 40 mins in presence of [gamma 33P]-ATP by radiometric scintillation counting assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA5158088 | B | Inhibition of recombinant full-length human NEK3 assessed as residual activity at 1 uM using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P]ATP by radiometric scintillation counting method relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA5158089 | B | Inhibition of recombinant full length human CaMK1gamma assessed as residual activity at 1 uM using KKLRRTLSFAEPG as substrate incubated for 40 mins in presence of [gamma-33ATP] by radiometric scintillation counting analysis relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA5158090 | B | Inhibition of recombinant human full length PKCalpha assessed as residual activity at 1 uM using histone H1 as substrate measured after 40 mins in presence of [gamma33P]ATP by radiometric scintillation counting method relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA5158091 | B | Inhibition of human full length recombinant CDK2/cyclinE assessed as residual activity at 1 uM using histone H1 as substrate incubated for 40 mins in presence of [gamma 33P]-ATP by radiometric scintillation counting assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 20. | ALA5158092 | B | Inhibition of recombinant full-length human Syk at 1 uM assessed as residual activity at 1 uM using poly(Glu, Tyr) 4:1 as substrate measured after 40 mins in presence of [gamma33P]ATP by radiometric scintillation counting method relative to control | Homo sapiens | 1 | single protein format | Scientific Literature |
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