| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5128818 | Functional | Antagonist activity at human alpha2A receptor stably expressed in CHO cells assessed as inhibition of adrenaline-induced response | Homo sapiens | 21 | ALA5126560 | cell-based format | Scientific Literature | |
| 2. | ALA5128819 | Functional | Antagonist activity at human alpha2C receptor stably expressed in CHO cells assessed as inhibition of adrenaline-induced response | Homo sapiens | 21 | ALA5126560 | cell-based format | Scientific Literature | |
| 3. | ALA5128820 | Binding | Selectivity ratio of Kb for antagonist activity at human alpha2A receptor stably expressed in CHO cells to Kb for antagonist activity at human alpha2C receptor stably expressed in CHO cells | Homo sapiens | 21 | ALA5126560 | cell-based format | Scientific Literature | |
| 4. | ALA5128821 | ADME | Clearance in human hepatocytes assessed per million cells at 1 uM | Homo sapiens | 21 | ALA5126560 | cell-based format | Scientific Literature | |
| 5. | ALA5128822 | ADME | Clearance in rat hepatocytes assessed per million cells at 1 uM | Rattus norvegicus | 21 | ALA5126560 | cell-based format | Scientific Literature | |
| 6. | ALA5128823 | Physicochemical | Lipophilicity, log D of compound at pH 7.4 | 21 | ALA5126560 | small-molecule physicochemical format | Scientific Literature | ||
| 7. | ALA5128824 | Physicochemical | Solubility of compound in pH 7.4 buffer at 1 uM | 20 | ALA5126560 | small-molecule physicochemical format | Scientific Literature |
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