| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5162518 | B | Binding affinity to His6-fused BRD9 (unknown origin) assessed as change in melting temperature at 100 uM incubated for 30 mins by thermal shift assay | Homo sapiens | 5 | ALA5154816 | single protein format | Scientific Literature | |
| 2. | ALA5162519 | B | Binding affinity to BRPF1 (unknown origin) assessed as change in melting temperature at 100 uM incubated for 30 mins by thermal shift assay | Homo sapiens | 5 | ALA5154816 | single protein format | Scientific Literature | |
| 3. | ALA5162520 | B | Binding affinity to BAZ2B (unknown origin) assessed as change in melting temperature at 100 uM incubated for 30 mins by thermal shift assay | Homo sapiens | 5 | ALA5154816 | single protein format | Scientific Literature | |
| 4. | ALA5162521 | T | Cytotoxicity against human HFL1 cells assessed as cell growth inhibition incubated for 72 hrs by Cell titre Glo-luminiscence cell viability assay | Homo sapiens | 2 | ALA5154816 | cell-based format | Scientific Literature | |
| 5. | ALA5162522 | B | Inhibition of C-terminal His6-tagged BRD4 BD1 (unknown origin) using H-YSGRGK(Ac)GGK(Ac)GLGK(Ac)-GGAK(Ac)RHRK-Biotin-OH as substrate incubated for 1 hrs by HTRF assay | Homo sapiens | 43 | ALA5154816 | single protein format | Scientific Literature | |
| 6. | ALA5162523 | B | Selectivity index, ratio of IC50 for BRD4 BD1 (unknown origin) to IC50 of BRD4 BD2 (unknown origin) | Homo sapiens | 43 | ALA5154816 | assay format | Scientific Literature | |
| 7. | ALA5162524 | B | Inhibition of C-terminal His6-tagged BRD4 BD2 (unknown origin) using H-YSGRGK(Ac)GGK(Ac)GLGK(Ac)-GGAK(Ac)RHRK-Biotin-OH as substrate incubated for 1 hrs by HTRF assay | Homo sapiens | 44 | ALA5154816 | single protein format | Scientific Literature | |
| 8. | ALA5162525 | B | Inhibition of C-terminal His6-tagged BRD3 BD2 (unknown origin) using H-YSGRGK(Ac)GGK(Ac)GLGK(Ac)-GGAK(Ac)RHRK-Biotin-OH as substrate incubated for 1 hrs by HTRF assay | Homo sapiens | 4 | ALA5154816 | single protein format | Scientific Literature | |
| 9. | ALA5162526 | B | Inhibition of C-terminal His6-tagged BRD2 BD2 (unknown origin) using H-YSGRGK(Ac)GGK(Ac)GLGK(Ac)-GGAK(Ac)RHRK-Biotin-OH as substrate incubated for 1 hrs by HTRF assay | Homo sapiens | 4 | ALA5154816 | single protein format | Scientific Literature | |
| 10. | ALA5162527 | B | Binding affinity to His6-fused BRD4 BD2 (unknown origin) assessed as change in melting temperature at 100 uM incubated for 30 mins by thermal shift assay | Homo sapiens | 5 | ALA5154816 | single protein format | Scientific Literature | |
| 11. | ALA5162528 | B | Binding affinity to His6-fused BRD3 BD2 (unknown origin) assessed as change in melting temperature at 100 uM incubated for 30 mins by thermal shift assay | Homo sapiens | 5 | ALA5154816 | single protein format | Scientific Literature | |
| 12. | ALA5162529 | B | Binding affinity to His6-fused BRD2 BD2 (unknown origin) assessed as change in melting temperature at 100 uM incubated for 30 mins by thermal shift assay | Homo sapiens | 5 | ALA5154816 | single protein format | Scientific Literature | |
| 13. | ALA5162530 | B | Binding affinity to His6-fused BRD3 BD1 (unknown origin) assessed as change in melting temperature at 100 uM incubated for 30 mins by thermal shift assay | Homo sapiens | 5 | ALA5154816 | single protein format | Scientific Literature | |
| 14. | ALA5162531 | B | Binding affinity to His6-fused BRD2 BD1 (unknown origin) assessed as change in melting temperature at 100 uM incubated for 30 mins by thermal shift assay | Homo sapiens | 5 | ALA5154816 | single protein format | Scientific Literature | |
| 15. | ALA5162532 | B | Binding affinity to His6-fused BRDT BD1 (unknown origin) assessed as change in melting temperature at 100 uM incubated for 30 mins by thermal shift assay | Homo sapiens | 5 | ALA5154816 | single protein format | Scientific Literature | |
| 16. | ALA5162533 | B | Binding affinity to CBP (unknown origin) assessed as change in melting temperature at 100 uM incubated for 30 mins by thermal shift assay | Homo sapiens | 5 | ALA5154816 | single protein format | Scientific Literature | |
| 17. | ALA5162534 | B | Inhibition of EP300 (unknown origin) assessed as change in melting temperature at 100 uM incubated for 30 mins by thermal shift assay | Homo sapiens | 5 | ALA5154816 | single protein format | Scientific Literature | |
| 18. | ALA5162535 | B | Binding affinity to CECR2 (unknown origin) assessed as change in melting temperature at 100 uM incubated for 30 mins by thermal shift assay | Homo sapiens | 5 | ALA5154816 | single protein format | Scientific Literature | |
| 19. | ALA5162536 | B | Binding affinity to PCAF (unknown origin) assessed as change in melting temperature at 100 uM incubated for 30 mins by thermal shift assay | Homo sapiens | 5 | ALA5154816 | single protein format | Scientific Literature | |
| 20. | ALA5162537 | B | Binding affinity to His6-fused BRD7 (unknown origin) assessed as change in melting temperature at 100 uM incubated for 30 mins by thermal shift assay | Homo sapiens | 5 | ALA5154816 | single protein format | Scientific Literature |
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