| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5116190 | B | Inhibition of human recombinant GST-tagged Clk1 (129 to 484 residues) expressed in Escherichia coli expression system at 100 nM using GRSRSRSRSRSRSRS peptide as substrate incubated for 15 mins in presence of ATP by phosphoimager analysis relative to control | Homo sapiens | 40 | assay format | Scientific Literature | ||
| 2. | ALA5116191 | B | Inhibition of human recombinant GST-tagged Clk1 (129 to 484 residues) expressed in Escherichia coli expression system using GRSRSRSRSRSRSRS peptide as substrate incubated for 15 mins in presence of ATP by phosphoimager analysis | Homo sapiens | 42 | assay format | Scientific Literature | ||
| 3. | ALA5116192 | B | Inhibition of human recombinant GST-tagged Clk2 expressed in Baculovirus expression system using GRSRSRSRSRSRSRS peptide as substrate incubated for 15 mins in presence of ATP by phosphoimager analysis | Homo sapiens | 5 | assay format | Scientific Literature | ||
| 4. | ALA5116193 | B | Inhibition of human recombinant GST-tagged Clk2 expressed in Baculovirus expression system at 0.25 uM using GRSRSRSRSRSRSRS peptide as substrate incubated for 15 mins in presence of ATP by phosphoimager analysis relative to control | Homo sapiens | 5 | assay format | Scientific Literature | ||
| 5. | ALA5116194 | B | Selectivity index, ratio of IC50 for human Clk2 to IC50 for human Clk1 by phosphoimager analysis | Homo sapiens | 5 | assay format | Scientific Literature | ||
| 6. | ALA5116195 | F | Antiproliferative activity against human T24 cells assessed as cell growth inhibition measured after 3 days by MTT assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 7. | ALA5116196 | B | Inhibition of human recombinant GST tagged/His-tagged full length CDK5/p25 expressed in Baculovirus expression system at 1 uM relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 8. | ALA5116197 | B | Inhibition of human recombinant GST tagged full length CSNK1D expressed in Baculovirus expression system at 1 uM relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 9. | ALA5116198 | B | Inhibition of CK2 (unknown origin) at 1 uM relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 10. | ALA5116199 | B | Inhibition of human recombinant GST-tagged full length CLK3 expressed in Baculovirus expression system at 1 uM relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 11. | ALA5116200 | B | Inhibition of human recombinant GST tagged full length CLK4 expressed in Baculovirus expression system at 1 uM relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 12. | ALA5116201 | B | Inhibition of human recombinant GST tagged full length DYRK1A expressed in Baculovirus expression system at 1 uM relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 13. | ALA5116202 | B | Inhibition of human recombinant GST tagged full length DYRK2 expressed in Escherichia coli expression system at 1 uM relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 14. | ALA5116203 | B | Inhibition of human recombinant GST tagged full length Haspin catalytic domain expressed in Baculovirus expression system at 1 uM relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 15. | ALA5116204 | B | Inhibition of human recombinant GST tagged HIPK1 expressed in Baculovirus expression system at 1 uM relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 16. | ALA5116205 | B | Inhibition of human recombinant His tagged full length Pim1 expressed in Baculovirus expression system at 1 uM relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 17. | ALA5116206 | B | Inhibition of human recombinant His tagged full length SRPK1 expressed in Baculovirus expression system at 1 uM relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 18. | ALA5116207 | B | Inhibition of human recombinant His tagged full length TRKB expressed in Baculovirus expression system at 1 uM relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 19. | ALA5116208 | B | Inhibition of human recombinant GST tagged full length CLK4 expressed in Baculovirus expression system at 1 uM | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 20. | ALA5116234 | B | Inhibition of human recombinant GST tagged full length MLCK2 expressed in Baculovirus expression system at 1 uM relative to control | Homo sapiens | 2 | assay format | Scientific Literature |
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