| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5142210 | Binding | Inhibition of His-tagged SMARCA4 (unknown origin) (1448 to 1575 residues) using biotinylated ARTKQTARKSTGG-K(Ac)-APR-K(Ac)-QLAT-K(Ac)-AAR-K(Ac)-SAPGG-K as substrate incubated for 10 mins by TR-FRET assay | Homo sapiens | 5 | ALA5137085 | single protein format | Scientific Literature | |
| 2. | ALA5142213 | Binding | Inhibition of BRD4 bromodomain 1 (unknown origin) by TR-FRET assay | Homo sapiens | 5 | ALA5137085 | single protein format | Scientific Literature | |
| 3. | ALA5142214 | Binding | Binding affinity to His6/FLAG-tagged SMARCA4 (unknown origin) by isothermal titration calorimetric assay | Homo sapiens | 5 | ALA5137085 | single protein format | Scientific Literature | |
| 4. | ALA5142215 | Binding | Binding affinity to human SMARCA4 (A1448 to S1575 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 5 | ALA5137085 | assay format | Scientific Literature | |
| 5. | ALA5142216 | Binding | Binding affinity to human SMARCA2 (S1337 to Q1486 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 5 | ALA5137085 | assay format | Scientific Literature | |
| 6. | ALA5142217 | Binding | Binding affinity to human PBRM1 bromodomain 5 (S645 to D766 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 5 | ALA5137085 | assay format | Scientific Literature | |
| 7. | ALA5142218 | Binding | Binding affinity to human PBRM1 bromodomain 2 (S178 to E291 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 5 | ALA5137085 | assay format | Scientific Literature | |
| 8. | ALA5142219 | Binding | Inhibition of SMARAC2 isoform B (unknown origin) expressed in U2OS cells co-expressed in NLS-ZsGreen incubated for 1 hrs by cellular target engagement assay | Homo sapiens | 5 | ALA5137085 | cell-based format | Scientific Literature | |
| 9. | ALA5142222 | Physicochemical | Kinetic solubility of compound | 2 | ALA5137085 | small-molecule physicochemical format | Scientific Literature | ||
| 10. | ALA5142223 | Physicochemical | Lipophilicity, LogD of compound | 2 | ALA5137085 | small-molecule physicochemical format | Scientific Literature | ||
| 11. | ALA5142224 | ADME | Clearance in mouse hepatocytes | Mus musculus | 1 | ALA5137085 | cell-based format | Scientific Literature | |
| 12. | ALA5142225 | ADME | Clearance in rat hepatocytes | Rattus norvegicus | 1 | ALA5137085 | cell-based format | Scientific Literature | |
| 13. | ALA5142226 | ADME | Clearance in human hepatocytes | Homo sapiens | 1 | ALA5137085 | cell-based format | Scientific Literature | |
| 14. | ALA5142227 | ADME | Inhibition of CYP3A4 (unknown origin) | Homo sapiens | 1 | ALA5137085 | single protein format | Scientific Literature | |
| 15. | ALA5142228 | ADME | Inhibition of CYP2C8 (unknown origin) | Homo sapiens | 1 | ALA5137085 | single protein format | Scientific Literature | |
| 16. | ALA5142229 | ADME | Inhibition of CYP2C19 (unknown origin) | Homo sapiens | 1 | ALA5137085 | single protein format | Scientific Literature | |
| 17. | ALA5142230 | ADME | Inhibition of CYP1A2 (unknown origin) | Homo sapiens | 1 | ALA5137085 | single protein format | Scientific Literature | |
| 18. | ALA5142231 | ADME | Inhibition of CYP2C9 (unknown origin) | Homo sapiens | 1 | ALA5137085 | single protein format | Scientific Literature | |
| 19. | ALA5142232 | ADME | Inhibition of CYP2D6 (unknown origin) | Homo sapiens | 1 | ALA5137085 | single protein format | Scientific Literature | |
| 20. | ALA5142233 | ADME | Protein binding in mouse plasma | Mus musculus | 1 | ALA5137085 | cell-free format | Scientific Literature |
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