# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA5158929 | B | Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate assessed as Kinact/Ki ratio and measured by colorimetric assay | Homo sapiens | 46 | ALA5154739 | single protein format | Scientific Literature | |
2. | ALA5158930 | B | Inhibition of TG2 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assay | Homo sapiens | 47 | ALA5154739 | single protein format | Scientific Literature | |
3. | ALA5158931 | B | Inhibition of GTP binding to TG2 (unknown origin) measured by GTP Gamma-S-FL BODIPY assay | Homo sapiens | 2 | ALA5154739 | single protein format | Scientific Literature | |
4. | ALA5158932 | B | Inhibition of TG1 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assay | Homo sapiens | 3 | ALA5154739 | single protein format | Scientific Literature | |
5. | ALA5158933 | B | Inhibition of TG6 (unknown origin) using Cbz-Glu(gamma-p-nitrophenyl ester)Gly (AL5) as substrate and measured by colorimetric assay | Homo sapiens | 3 | ALA5154739 | single protein format | Scientific Literature | |
6. | ALA5158934 | B | Inhibition of TG3 (unknown origin) using peptidic FRET quenched probe A101 as substrate and measured by fluorescence-based assay | Homo sapiens | 3 | ALA5154739 | single protein format | Scientific Literature | |
7. | ALA5158935 | B | Inhibition of FXIIIa (unknown origin) using peptidic FRET quenched probe A101 as substrate and measured by fluorescence-based assay | Homo sapiens | 3 | ALA5154739 | single protein format | Scientific Literature | |
8. | ALA5158936 | A | Half-life in plasma (unknown origin) | Not specified | 2 | ALA5154739 | cell-free format | Scientific Literature | |
9. | ALA5158937 | A | Half-life in hepatocytes (unknown origin) | Not specified | 2 | ALA5154739 | cell-based format | Scientific Literature | |
10. | ALA5158938 | A | Intrinsic clearance in hepatocytes (unknown origin) assessed per million cells | Not specified | 2 | ALA5154739 | cell-based format | Scientific Literature | |
11. | ALA5158939 | A | Plasma protein binding (unknown origin) | Not specified | 2 | ALA5154739 | cell-free format | Scientific Literature | |
12. | ALA5158940 | A | Plasma protein binding (unknown origin) assessed as drug recovery | Not specified | 2 | ALA5154739 | cell-free format | Scientific Literature | |
13. | ALA5158941 | A | Permeability coefficient of compound by PAMPA assay | 2 | ALA5154739 | assay format | Scientific Literature | ||
14. | ALA5158942 | A | Apparent permeability from apical to basolateral side in dog MDCK-MDR1 cells | Canis lupus familiaris | 2 | ALA5154739 | cell-based format | Scientific Literature | |
15. | ALA5158943 | A | Apparent permeability from basolateral to apical side in dog MDCK-MDR1 cells | Canis lupus familiaris | 2 | ALA5154739 | cell-based format | Scientific Literature | |
16. | ALA5158944 | A | Efflux ratio of apparent permeability in dog MDCK-MDR1 cells | Canis lupus familiaris | 2 | ALA5154739 | cell-based format | Scientific Literature | |
17. | ALA5158945 | A | Substrate activity at P-gp in dog MDCK cells assessed as apparent permeability across apical to basolateral membrane | Canis lupus familiaris | 2 | ALA5154739 | cell-based format | Scientific Literature | |
18. | ALA5158946 | A | Substrate activity at P-gp in dog MDCK cells assessed as apparent permeability across basolateral to apical membrane | Canis lupus familiaris | 2 | ALA5154739 | cell-based format | Scientific Literature | |
19. | ALA5158947 | A | Substrate activity at P-gp in dog MDCK cells assessed as efflux ratio | Canis lupus familiaris | 2 | ALA5154739 | cell-based format | Scientific Literature | |
20. | ALA5158948 | F | Anti-invasion activity against human SCC-13 cells assessed as inhibition of invasion incubated for 18 hrs by matrigel trans well plate assay | Homo sapiens | 6 | ALA5154739 | cell-based format | Scientific Literature |