| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5159712 | B | Inhibition of N-terminal His/GST-tagged human LSD1 (172 to 852 residues) expressed in expressed in baculovirus infected insect cells using biotinylated H3K4Me2 peptide as substrate by TR-FRET assay | Homo sapiens | 29 | ALA5154758 | cell-based format | Scientific Literature | |
| 2. | ALA5159713 | B | Inhibition of recombinant human full length LSD2 using biotinylated H3K4Me2 peptide as substrate by TR-FRET assay | Homo sapiens | 24 | ALA5154758 | single protein format | Scientific Literature | |
| 3. | ALA5159714 | B | Inhibition of human recombinant MAO-A expressed in baculovirus infected BTI insect cells using luminogenic MAO substrate incubated for 1 hr by luciferin-based luminescence assay | Homo sapiens | 26 | ALA5154758 | cell-based format | Scientific Literature | |
| 4. | ALA5159715 | B | Inhibition of human recombinant MAO-B expressed in baculovirus infected BTI insect cells using luminogenic MAO substrate incubated for 1 hr by luciferin-based luminescence assay | Homo sapiens | 26 | ALA5154758 | cell-based format | Scientific Literature | |
| 5. | ALA5159716 | B | Selectivity index, ratio of IC50 for inhibition of recombinant human full length LSD2 to IC50 for inhibition of N-terminal His/GST-tagged human LSD1 (172 to 852 residues) expressed in baculovirus infected insect cells | Homo sapiens | 24 | ALA5154758 | cell-based format | Scientific Literature | |
| 6. | ALA5159717 | F | Upregulation of CD86 expression in human MV4-11 cells assessed as fold change in CD86 expression at IC50 incubated for 24 hrs by qRT-PCR analysis relative to control | Homo sapiens | 9 | ALA5154758 | cell-based format | Scientific Literature | |
| 7. | ALA5159718 | F | Antiproliferative activity against human MV4-11 cells assessed as inhibition of cell growth incubated for 240 hrs by MTS assay | Homo sapiens | 9 | ALA5154758 | cell-based format | Scientific Literature | |
| 8. | ALA5159719 | F | Antiproliferative activity against human RPMI-8226 cells assessed as inhibition of cell growth incubated for 240 hrs by MTS assay | Homo sapiens | 4 | ALA5154758 | cell-based format | Scientific Literature |
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