# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA5115899 | B | Irreversible inhibition of Trypanosoma brucei rhodesiense rhodesain assessed as inhibition constant using Cbz-Phe-Arg-AMC as fluorogenic substrate by fluorometric assay | Trypanosoma brucei rhodesiense | 30 | single protein format | Scientific Literature | ||
2. | ALA5115900 | B | Irreversible inhibition of Trypanosoma brucei rhodesiense rhodesain assessed as Kinact using Cbz-Phe-Arg-AMC as fluorogenic substrate by fluorometric assay | Trypanosoma brucei rhodesiense | 20 | single protein format | Scientific Literature | ||
3. | ALA5115901 | B | Irreversible inhibition of Trypanosoma brucei rhodesiense rhodesain assessed as second order rate constant using Cbz-Phe-Arg-AMC as fluorogenic substrate by fluorometric assay | Trypanosoma brucei rhodesiense | 20 | single protein format | Scientific Literature | ||
4. | ALA5115902 | B | Irreversible inhibition of human Cathepsin L assessed as inhibition constant using Cbz-Phe-Arg-AMC as fluorogenic substrate by fluorometric assay | Homo sapiens | 9 | single protein format | Scientific Literature | ||
5. | ALA5115903 | B | Irreversible inhibition of human Cathepsin L assessed as Kinact using Cbz-Phe-Arg-AMC as fluorogenic substrate by fluorometric assay | Homo sapiens | 10 | single protein format | Scientific Literature | ||
6. | ALA5115904 | B | Irreversible inhibition of human Cathepsin L assessed as second order rate constant using Cbz-Phe-Arg-AMC as fluorogenic substrate by fluorometric assay | Homo sapiens | 10 | single protein format | Scientific Literature | ||
7. | ALA5115905 | B | Irreversible inhibition of human Cathepsin B assessed as inhibition constant using Cbz-Phe-Arg-AMC as fluorogenic substrate by fluorometric assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
8. | ALA5115906 | B | Irreversible inhibition of human Cathepsin B assessed as Kinact using Cbz-Phe-Arg-AMC as fluorogenic substrate by fluorometric assay | Homo sapiens | 10 | single protein format | Scientific Literature | ||
9. | ALA5115907 | B | Irreversible inhibition of human Cathepsin B assessed as second order rate constant using Cbz-Phe-Arg-AMC as fluorogenic substrate by fluorometric assay | Homo sapiens | 10 | single protein format | Scientific Literature | ||
10. | ALA5115913 | B | Inhibition of human 20S proteasome trypsin-like activity at 11 uM using Boc-Leu-Arg-Arg-AMC as fluorogenic substrate by fluorometric assay | Homo sapiens | 7 | protein complex format | Scientific Literature | ||
11. | ALA5115914 | B | Inhibition of human 20S proteasome caspase-like activity at 11 uM using Cbz-Leu-Leu-Glu-AMC as fluorogenic substrate by fluorometric assay | Homo sapiens | 7 | protein complex format | Scientific Literature | ||
12. | ALA5115915 | B | Inhibition of human 20S proteasome chymotrypsin-like activity at 11 uM using Succ-Leu-Leu-Val-Tyr-AMC as fluorogenic substrate by fluorometric assay | Homo sapiens | 7 | protein complex format | Scientific Literature | ||
13. | ALA5115916 | B | Inhibition of Dengue virus NS2B-NS3 protease at 11 uM using Boc-Gly-Arg-Arg-AMC as fluorogenic substrate by fluorometric assay | Dengue virus | 7 | single protein format | Scientific Literature | ||
14. | ALA5115918 | B | Irreversible inhibition of Trypanosoma brucei rhodesiense rhodesain assessed as no recovery of enzyme activity preincubated for 30 mins followed by substrate addition using Cbz-Phe-Arg-AMC as fluorogenic substrate by fluorometric 100-fold dilution assay | Trypanosoma brucei rhodesiense | 5 | single protein format | Scientific Literature |