| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5129799 | B | Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equation analysis | Homo sapiens | 27 | ALA5126603 | cell membrane format | Scientific Literature | |
| 2. | ALA5129800 | B | Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation analysis | Homo sapiens | 10 | ALA5126603 | cell membrane format | Scientific Literature | |
| 3. | ALA5129814 | A | Metabolic stability in human plasma assessed as half life at 5 uM measured upto 120 mins by LC-MS/MS analysis | Homo sapiens | 8 | ALA5126603 | cell-free format | Scientific Literature | |
| 4. | ALA5129815 | A | Metabolic stability in rat plasma assessed as half life at 5 uM measured upto 120 mins by LC-MS/MS analysis | Rattus norvegicus | 8 | ALA5126603 | cell-free format | Scientific Literature | |
| 5. | ALA5129841 | F | Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contraction in presence of propranolol | Cavia porcellus | 8 | ALA5126603 | tissue-based format | Scientific Literature | |
| 6. | ALA5129842 | F | Invivo bifunctional antagonist activity at muscarinic M3 receptor /agonist activity at beta-2 adrenoceptor in Dunkin-Hartley guinea pig trachea assessed as time duration for inhibition of carbachol induced contraction measured upto 4 hrs | Cavia porcellus | 8 | ALA5126603 | tissue-based format | Scientific Literature | |
| 7. | ALA5129843 | F | Invivo agonist beta2 adrenoceptor activity in Dunkin-Hartley guinea pig trachea assessed as histamine induced contraction | Cavia porcellus | 8 | ALA5126603 | tissue-based format | Scientific Literature | |
| 8. | ALA5129844 | F | Invivo bifunctional antagonist activity at muscarinic M3 receptor /agonist activity at beta-2 adrenoceptor in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contraction | Cavia porcellus | 8 | ALA5126603 | tissue-based format | Scientific Literature |
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