| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5107056 | B | Displacement of [125I]-NDP-alpha-MSH from human MC1R expressed in HEK2936E cell membrane measured after 16 to 23 hrs by 1450 microbeta trilux scintillation proximity assay | Homo sapiens | 31 | cell membrane format | Scientific Literature | ||
| 2. | ALA5107057 | B | Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK2936E cell membrane measured after 16 to 23 hrs by 1450 microbeta trilux scintillation proximity assay | Homo sapiens | 31 | cell membrane format | Scientific Literature | ||
| 3. | ALA5107058 | B | Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK2936E cell membrane measured after 16 to 23 hrs by 1450 microbeta trilux scintillation proximity assay | Homo sapiens | 31 | cell membrane format | Scientific Literature | ||
| 4. | ALA5107059 | F | Agonist activity at human MC1R expressed in HEK2936E cells assessed as cAMP production in presence of IBMX by time resolved fluorescence assay | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 5. | ALA5107060 | F | Agonist activity at human MC3R expressed in HEK2936E cells assessed as cAMP production in presence of IBMX by time resolved fluorescence assay | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 6. | ALA5107061 | F | Antagonist activity at human MC4R expressed in HEK2936E cells assessed as cAMP production in presence of IBMX by time resolved fluorescence assay | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 7. | ALA5107062 | F | Agonist activity at human MC5R expressed in HEK2936E cells assessed as cAMP production in presence of IBMX by time resolved fluorescence assay | Homo sapiens | 31 | cell-based format | Scientific Literature | ||
| 8. | ALA5107063 | B | Selectivity ratio of Ki for human MC3R to Ki for human MC1R | Homo sapiens | 31 | assay format | Scientific Literature | ||
| 9. | ALA5107064 | B | Selectivity ratio of Ki for human MC4R to Ki for human MC1R | Homo sapiens | 31 | assay format | Scientific Literature | ||
| 10. | ALA5107065 | B | Selectivity ratio of EC50 for human MC3R to EC50 for human MC1R | Homo sapiens | 31 | assay format | Scientific Literature | ||
| 11. | ALA5107066 | B | Selectivity ratio of EC50 for human MC4R to EC50 for human MC1R | Homo sapiens | 31 | assay format | Scientific Literature |
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