| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5217581 | Binding | Inhibition of N-terminal his-tagged human recombinant BCAT1 expressed in Escherichia coli BL21(DE3) cells using leucine and alpha-KG as substrate in presence of NADH by fluorescence assay | Homo sapiens | 39 | ALA5214979 | cell-based format | Scientific Literature | |
| 2. | ALA5217582 | Binding | Inhibition of human recombinant BCAT2 using leucine and alpha-KG as substrate in presence of NADH by fluorescence assay | Homo sapiens | 27 | ALA5214979 | single protein format | Scientific Literature | |
| 3. | ALA5217583 | ADME | Apparent permeability of the compound from apical to basolateral side in human Caco-2 cells incubated for 2 hrs by LC-MS/MS analysis | Homo sapiens | 15 | ALA5214979 | cell-based format | Scientific Literature | |
| 4. | ALA5217584 | ADME | Efflux ratio of apparent permeability in human Caco-2 cells incubated for 2 hrs by LC-MS/MS analysis | Homo sapiens | 16 | ALA5214979 | cell-based format | Scientific Literature | |
| 5. | ALA5217600 | Functional | Upregulation of BCAA expression in human U-87 MG cells | Homo sapiens | 4 | ALA5214979 | cell-based format | Scientific Literature | |
| 6. | ALA5217601 | Functional | Upregulation of BCAA expression in human MDA-MB-231 cells | Homo sapiens | 3 | ALA5214979 | cell-based format | Scientific Literature |
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