| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5218148 | B | Inhibition of BRD4 BD2 (unknown origin) measured by TR-FRET assay | Homo sapiens | 45 | ALA5214999 | single protein format | Scientific Literature | |
| 2. | ALA5218149 | B | Inhibition of BRD4 BD1 (unknown origin) measured by TR-FRET assay | Homo sapiens | 45 | ALA5214999 | single protein format | Scientific Literature | |
| 3. | ALA5218150 | B | Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assay | Homo sapiens | 29 | ALA5214999 | tissue-based format | Scientific Literature | |
| 4. | ALA5218151 | P | Lipophilicity, logD of compound at pH 7.4 by Chromatography | 37 | ALA5214999 | small-molecule physicochemical format | Scientific Literature | ||
| 5. | ALA5218155 | A | Artificial membrane permeability of the compound | 33 | ALA5214999 | assay format | Scientific Literature | ||
| 6. | ALA5218157 | P | Solubility of the compound at pH 6.5 in fast state simulated intestinal fluid incubated for 16 hrs by HPLC analysis | 5 | ALA5214999 | small-molecule physicochemical format | Scientific Literature | ||
| 7. | ALA5218158 | A | Intrinsic clearance in rat hepatocytes after 60 mins by LC-MS/MS analysis | Rattus norvegicus | 9 | ALA5214999 | cell-based format | Scientific Literature | |
| 8. | ALA5218160 | A | Intrinsic clearance in human hepatocytes measured after 120 mins by LC-MS/MS analysis | Homo sapiens | 9 | ALA5214999 | cell-based format | Scientific Literature | |
| 9. | ALA5218168 | A | Clearance in Wistar Han rat blood at 2.9 mg/kg, po or 2.1 mg/kg, iv measured upto 24 hrs by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA5214999 | organism-based format | Scientific Literature | |
| 10. | ALA5218169 | A | Volume of distribution at steady state in Wistar Han rat at 2.9 mg/kg, po or 2.1 mg/kg, iv measured upto 24 hrs by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA5214999 | organism-based format | Scientific Literature | |
| 11. | ALA5218170 | A | Half-life in Wistar Han rat at 2.9 mg/kg, po or 2.1 mg/kg, iv measured upto 24 hrs by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA5214999 | organism-based format | Scientific Literature | |
| 12. | ALA5218171 | A | Oral bioavailability in Wistar Han rat at 2.9 mg/kg measured upto 24 hrs by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA5214999 | organism-based format | Scientific Literature |
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