| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA5218411 | F | Induction of adipogenesis in differentiated human BMMSC cells assessed as fold increase in adiponectin level at 30 uM in presence of IDX by ELISA relative to control | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 2. | ALA5218413 | F | Induction of adipogenesis in differentiated human BMMSC cells assessed as fold increase in adiponectin level in presence of IDX by ELISA | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 3. | ALA5218414 | F | Induction of adipogenesis in differentiated human BMMSC cells assessed as increase in number and size of lipid droplets at 30 uM in presence of IDX by Oil red O staining based inverted microscope analysis | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 4. | ALA5218415 | B | Displacement of fluormone pan-PPARgreen from PPARalpha (unknown origin) at 30 uM by TR-FRET based competitive binding assay relative to control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 5. | ALA5218416 | B | Displacement of fluormone pan-PPARgreen from PPARgamma (unknown origin) at 30 uM by TR-FRET based competitive binding assay relative to control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 6. | ALA5218417 | B | Displacement of fluormone pan-PPARgreen from PPARdelta (unknown origin) at 30 uM by TR-FRET based competitive binding assay relative to control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 7. | ALA5218421 | B | Binding affinity to PPARalpha (unknown origin) assessed as inhibition constant by Cheng-Prusoff equation analysis | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 8. | ALA5218422 | B | Binding affinity to PPARgamma (unknown origin) assessed as inhibition constant by Cheng-Prusoff equation analysis | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 9. | ALA5218423 | B | Binding affinity to PPARdelta (unknown origin) assessed as inhibition constant by Cheng-Prusoff equation analysis | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 10. | ALA5218424 | B | Partial agonist activity at PPARgamma in human BMMSC cells assessed as inhibition of pioglitazone-induced adiponectin synthesis measured after 5 days by ELISA | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 11. | ALA5218425 | B | Partial agonist activity at PPARalpha (unknown origin) assessed as increase in PRIP/RAP250 coactivator peptide requirement by Lanthascreen TR-FRET assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 12. | ALA5218426 | B | Partial agonist activity at PPARgamma (unknown origin) assessed as increase in fluorescein labeled PRIP/RAP250 coactivator peptide requirement by Lanthascreen TR-FRET assay | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 13. | ALA5218429 | B | Partial agonist activity at PPARgamma (unknown origin) assessed as increase in fluorescein labeled SMRT corepressor peptide requirement by Lanthascreen TR-FRET assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 14. | ALA5218430 | B | Partial agonist activity at PPARalpha (unknown origin) assessed as increase in fluorescein labeled SMRT corepressor peptide requirement by Lanthascreen TR-FRET assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 15. | ALA5218431 | B | Partial agonist activity at PPARdelta (unknown origin) assessed as increase in fluorescein labeled SMRT corepressor peptide requirement by Lanthascreen TR-FRET assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 16. | ALA5218432 | B | Partial agonist activity at PPARdelta (unknown origin) assessed as increase in fluorescein labeled PRIP/RAP250 coactivator peptide requirement by Lanthascreen TR-FRET assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 17. | ALA5218434 | B | Agonist activity at RXRalpha-LBD (unknown origin) assessed as transactivation by measuring increase in fluorescein-labelled coactivator PGC-1alpha peptide recruitment by Lanthascreen TR-FRET | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 18. | ALA5218435 | B | Agonist activity at RXRbeta-LBD (unknown origin) assessed as transactivation by measuring increase in fluorescein-labelled coactivator D22 peptide recruitment by Lanthascreen TR-FRET assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 19. | ALA5218436 | B | Agonist activity at FXR (unknown origin) assessed as transactivation by measuring increase in fluorescein-labelled coactivator SRC-2 peptide recruitment by Lanthascreen TR-FRET assay | Homo sapiens | 2 | single protein format | Scientific Literature |
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